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Compound Detail

CHEMBL6005633

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CC1CN(CCS(C)(=O)=O)CCC(O[C@@H]2[C@H](C)O[C@@H](O[C@@H]3[C@H](C)O[C@@H](O[C@H]4CC[C@@]5(C)C(CCC6C5C[C@H](O)[C@]5(C)[C@@H](C7=CC(=O)OC7)CC[C@]65O)C4)C[C@@H]3O)C[C@@H]2O)O1

Basic Information

ChEMBL ID CHEMBL6005633
Phase Preclinical
Structure Type MOL
InChI Key RXELIABRBGFTHS-AJOSXQTQSA-N
4
Targets
4
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

870.1
MW (Da)
2.84
ALogP
15
HBA
4
HBD
200.0
PSA (Ų)
0.18
QED
2
Ro5 Violations
10
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C44H71NO14S
MW 870.11
Aromatic Rings 0
Heavy Atoms 60
NP-Likeness 1.56

Activity Summary

Ki 4 meas. best 7.61

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Sodium/potassium-transporting ATPase subunit alpha-2/beta-3
CHEMBL6066562
Ki 7.61 7.61 24.7 1
Sodium/potassium-transporting ATPase subunit alpha-2/beta-2
CHEMBL6066561
Ki 7.5 7.5 31.7 1
Sodium/potassium-transporting ATPase subunit alpha-2/beta-1
CHEMBL6066560
Ki 7.31 7.31 49.2 1
Sodium/potassium-transporting ATPase subunit alpha-1/beta-1
CHEMBL6066559
Ki 6.33 6.33 464.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine