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Compound Detail

CHEMBL72170

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N#Cc1ccc(NC(=S)NS(=O)(=O)Cc2c(Cl)cccc2Cl)cc1

Basic Information

ChEMBL ID CHEMBL72170
Phase Preclinical
Structure Type MOL
InChI Key VVDXAJUSAOXLLI-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

400.3
MW (Da)
3.68
ALogP
4
HBA
2
HBD
82.0
PSA (Ų)
0.77
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C15H11Cl2N3O2S2
MW 400.31
Aromatic Rings 2
Heavy Atoms 24
NP-Likeness -1.89

Activity Summary

IC50 1 meas. best 4.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human immunodeficiency virus 1
CHEMBL378
IC50 4.0 4.0 100000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Human immunodeficiency virus 1 IC50 = 100000.0 nM 4.0 Compound potency to achieve protection of MT-4 cells from HIV-1 cytopathicity 11527703

Literature References

PubMed DOI Target Context # Activities
11527703 10.1016/s0960-894x(01)00410-3 Human immunodeficiency virus 1 1

Data from ChEMBL 36 via Core Engine