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Compound Detail

CHEMBL92308

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O=C1c2cccn2-c2ccccc2OC1(CC1CC1)c1ccccc1

Basic Information

ChEMBL ID CHEMBL92308
Phase Preclinical
Structure Type MOL
InChI Key VUBUOKJQMWJAGL-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

329.4
MW (Da)
4.75
ALogP
3
HBA
0
HBD
31.2
PSA (Ų)
0.69
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H19NO2
MW 329.40
Aromatic Rings 3
Heavy Atoms 25

Activity Summary

IC50 1 meas. best 4.93

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
CEM-SS
CHEMBL614548
IC50 4.93 4.93 11800.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
CEM-SS IC50 = 11800.0 nM 4.93 Cytotoxic concentration against 50% survival of uninfected untreated control CEM... 8709096

Literature References

PubMed DOI Target Context # Activities
8709096 10.1021/jm950702c Human immunodeficiency virus type 1 reverse transcriptase 1
8709096 10.1021/jm950702c CEM-SS 1

Data from ChEMBL 36 via Core Engine