Assay Detail
Functional
CHEMBL1613827
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response cell-based assay to measure STAT1 inhibition. (Class of assay: confirmatory) [Related pubchem assays: 1263, 920, 862, 1303, 1310 ]
53
Total Activities
53
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Signal transducer and activator of transcription 1-alpha/beta (CHEMBL6101) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 53 | 4.93 | 5.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1299252 | — | — | 1 | 5.46 |
| CHEMBL1574527 | — | — | 1 | 5.45 |
| CHEMBL1424535 | — | — | 1 | 5.37 |
| CHEMBL1324820 | — | — | 1 | 5.36 |
| CHEMBL1518821 | — | — | 1 | 5.35 |
| CHEMBL1374466 | — | — | 1 | 5.28 |
| CHEMBL3195771 | — | — | 1 | 5.20 |
| CHEMBL1502512 | — | — | 1 | 5.17 |
| CHEMBL1326850 | — | — | 1 | 5.10 |
| CHEMBL1541307 | — | — | 1 | 5.07 |
| CHEMBL1444667 | — | — | 1 | 5.03 |
| CHEMBL1420733 | — | — | 1 | 5.03 |
| CHEMBL1607286 | — | — | 1 | 5.02 |
| CHEMBL1492648 | — | — | 1 | 5.00 |
| CHEMBL1429929 | — | — | 1 | 4.99 |
| CHEMBL1447780 | — | — | 1 | 4.98 |
| CHEMBL1986725 | — | — | 1 | 4.98 |
| CHEMBL1370681 | — | — | 1 | 4.97 |
| CHEMBL1465899 | — | — | 1 | 4.96 |
| CHEMBL1479604 | — | — | 1 | 4.94 |
| CHEMBL1601512 | — | — | 1 | 4.93 |
| CHEMBL1487321 | — | — | 1 | 4.93 |
| CHEMBL1375338 | — | — | 1 | 4.92 |
| CHEMBL1462729 | — | — | 1 | 4.88 |
| CHEMBL1354211 | — | — | 1 | 4.87 |
| CHEMBL1382249 | — | — | 1 | 4.85 |
| CHEMBL1461002 | — | — | 1 | 4.83 |
| CHEMBL1568022 | — | — | 1 | 4.77 |
| CHEMBL1371761 | — | — | 1 | 4.77 |
| CHEMBL1574403 | — | — | 1 | 4.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1299252 | — | IC50 | = | 3467.0 | nM | 5.46 |
| CHEMBL1574527 | — | IC50 | = | 3517.0 | nM | 5.45 |
| CHEMBL1424535 | — | IC50 | = | 4239.0 | nM | 5.37 |
| CHEMBL1324820 | — | IC50 | = | 4363.0 | nM | 5.36 |
| CHEMBL1518821 | — | IC50 | = | 4423.0 | nM | 5.35 |
| CHEMBL1374466 | — | IC50 | = | 5195.0 | nM | 5.28 |
| CHEMBL3195771 | — | IC50 | = | 6371.0 | nM | 5.20 |
| CHEMBL1502512 | — | IC50 | = | 6702.0 | nM | 5.17 |
| CHEMBL1326850 | — | IC50 | = | 7874.0 | nM | 5.10 |
| CHEMBL1541307 | — | IC50 | = | 8427.0 | nM | 5.07 |
| CHEMBL1444667 | — | IC50 | = | 9254.0 | nM | 5.03 |
| CHEMBL1420733 | — | IC50 | = | 9385.0 | nM | 5.03 |
| CHEMBL1607286 | — | IC50 | = | 9576.0 | nM | 5.02 |
| CHEMBL1492648 | — | IC50 | = | 9973.0 | nM | 5.00 |
| CHEMBL1429929 | — | IC50 | = | 10160.0 | nM | 4.99 |
| CHEMBL1447780 | — | IC50 | = | 10450.0 | nM | 4.98 |
| CHEMBL1986725 | — | IC50 | = | 10480.0 | nM | 4.98 |
| CHEMBL1370681 | — | IC50 | = | 10650.0 | nM | 4.97 |
| CHEMBL1465899 | — | IC50 | = | 11090.0 | nM | 4.96 |
| CHEMBL1479604 | — | IC50 | = | 11420.0 | nM | 4.94 |
| CHEMBL1601512 | — | IC50 | = | 11850.0 | nM | 4.93 |
| CHEMBL1487321 | — | IC50 | = | 11870.0 | nM | 4.93 |
| CHEMBL1375338 | — | IC50 | = | 12050.0 | nM | 4.92 |
| CHEMBL1462729 | — | IC50 | = | 13330.0 | nM | 4.88 |
| CHEMBL1354211 | — | IC50 | = | 13500.0 | nM | 4.87 |
| CHEMBL1382249 | — | IC50 | = | 14050.0 | nM | 4.85 |
| CHEMBL1461002 | — | IC50 | = | 14840.0 | nM | 4.83 |
| CHEMBL1568022 | — | IC50 | = | 16860.0 | nM | 4.77 |
| CHEMBL1371761 | — | IC50 | = | 16820.0 | nM | 4.77 |
| CHEMBL1574403 | — | IC50 | = | 16900.0 | nM | 4.77 |
| CHEMBL1578386 | — | IC50 | = | 17830.0 | nM | 4.75 |
| CHEMBL1340469 | — | IC50 | = | 18500.0 | nM | 4.73 |
| CHEMBL1352434 | — | IC50 | = | 21180.0 | nM | 4.67 |
| CHEMBL1539189 | — | IC50 | = | 21140.0 | nM | 4.67 |
| CHEMBL1525358 | — | IC50 | = | 21680.0 | nM | 4.66 |
| CHEMBL1545160 | — | IC50 | = | 23610.0 | nM | 4.63 |
| CHEMBL1492504 | — | IC50 | = | 26580.0 | nM | 4.58 |
| CHEMBL1328462 | — | IC50 | = | 31010.0 | nM | 4.51 |
| CHEMBL1389279 | — | IC50 | = | 42630.0 | nM | 4.37 |
| CHEMBL1378851 | — | IC50 | = | 47300.0 | nM | 4.33 |
| CHEMBL1444859 | — | IC50 | > | 18600.0 | nM | - |
| CHEMBL1518620 | — | IC50 | > | 55700.0 | nM | - |
| CHEMBL1308733 | — | IC50 | > | 55700.0 | nM | - |
| CHEMBL1606613 | — | IC50 | > | 18600.0 | nM | - |
| CHEMBL1360505 | — | IC50 | > | 55700.0 | nM | - |
| CHEMBL1447505 | — | IC50 | > | 55700.0 | nM | - |
| CHEMBL1385084 | — | IC50 | > | 55700.0 | nM | - |
| CHEMBL1335610 | — | IC50 | > | 18600.0 | nM | - |
| CHEMBL1304647 | — | IC50 | > | 55700.0 | nM | - |
| CHEMBL1329658 | — | IC50 | > | 55700.0 | nM | - |