Assay Detail
Binding
CHEMBL1613873
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: LYP1 Fluorescent Assay using OMFP substrate for In Vitro dose response studies. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1779, AID1784, AID435024]
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 22 (CHEMBL2889) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 5.16 | 5.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1320181 | — | — | 1 | 5.88 |
| CHEMBL1533230 | — | — | 1 | 5.37 |
| CHEMBL1424694 | — | — | 1 | 5.34 |
| CHEMBL1438889 | — | — | 1 | 5.33 |
| CHEMBL2000167 | — | — | 1 | 5.32 |
| CHEMBL1426096 | — | — | 1 | 5.31 |
| CHEMBL1492305 | — | — | 1 | 5.21 |
| CHEMBL1371816 | — | — | 1 | 5.08 |
| CHEMBL1439815 | — | — | 1 | 4.77 |
| CHEMBL1443268 | — | — | 1 | 4.73 |
| CHEMBL1417070 | — | — | 1 | 4.40 |
| CHEMBL1701224 | — | — | 1 | - |
| CHEMBL1445488 | — | — | 1 | - |
| CHEMBL1464805 | — | — | 1 | - |
| CHEMBL1993612 | — | — | 1 | - |
| CHEMBL2001743 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1320181 | — | IC50 | = | 1303.12 | nM | 5.88 |
| CHEMBL1533230 | — | IC50 | = | 4283.08 | nM | 5.37 |
| CHEMBL1424694 | — | IC50 | = | 4539.51 | nM | 5.34 |
| CHEMBL1438889 | — | IC50 | = | 4659.16 | nM | 5.33 |
| CHEMBL2000167 | — | IC50 | = | 4829.18 | nM | 5.32 |
| CHEMBL1426096 | — | IC50 | = | 4852.77 | nM | 5.31 |
| CHEMBL1492305 | — | IC50 | = | 6142.23 | nM | 5.21 |
| CHEMBL1371816 | — | IC50 | = | 8283.5 | nM | 5.08 |
| CHEMBL1439815 | — | IC50 | = | 16844.96 | nM | 4.77 |
| CHEMBL1443268 | — | IC50 | = | 18785.38 | nM | 4.73 |
| CHEMBL1417070 | — | IC50 | = | 39932.83 | nM | 4.40 |
| CHEMBL1701224 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1445488 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1464805 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1993612 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL2001743 | — | IC50 | > | 99000.0 | nM | - |