Assay Detail
Functional
CHEMBL1614145
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: HTS HePTP Fluorescent Assay using OMFP substrate for In Vitro dose response studies. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1059, AID1077, AID1784, AID2068, AID2085, AID435032, AID521]
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 7 (CHEMBL2219) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 4.96 | 5.32 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1426096 | — | — | 1 | 5.32 |
| CHEMBL1320181 | — | — | 1 | 5.31 |
| CHEMBL2000167 | — | — | 1 | 5.29 |
| CHEMBL1438889 | — | — | 1 | 5.25 |
| CHEMBL1424694 | — | — | 1 | 5.22 |
| CHEMBL1371816 | — | — | 1 | 5.10 |
| CHEMBL1443268 | — | — | 1 | 5.06 |
| CHEMBL1492305 | — | — | 1 | 4.61 |
| CHEMBL1533230 | — | — | 1 | 4.54 |
| CHEMBL1417070 | — | — | 1 | 4.43 |
| CHEMBL1464805 | — | — | 1 | 4.42 |
| CHEMBL1701224 | — | — | 1 | - |
| CHEMBL1445488 | — | — | 1 | - |
| CHEMBL1993612 | — | — | 1 | - |
| CHEMBL1439815 | — | — | 1 | - |
| CHEMBL2001743 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1426096 | — | IC50 | = | 4777.0 | nM | 5.32 |
| CHEMBL1320181 | — | IC50 | = | 4940.0 | nM | 5.31 |
| CHEMBL2000167 | — | IC50 | = | 5119.0 | nM | 5.29 |
| CHEMBL1438889 | — | IC50 | = | 5640.0 | nM | 5.25 |
| CHEMBL1424694 | — | IC50 | = | 6060.0 | nM | 5.22 |
| CHEMBL1371816 | — | IC50 | = | 7880.0 | nM | 5.10 |
| CHEMBL1443268 | — | IC50 | = | 8800.0 | nM | 5.06 |
| CHEMBL1492305 | — | IC50 | = | 24557.0 | nM | 4.61 |
| CHEMBL1533230 | — | IC50 | = | 28580.0 | nM | 4.54 |
| CHEMBL1417070 | — | IC50 | = | 37467.0 | nM | 4.43 |
| CHEMBL1464805 | — | IC50 | = | 37880.0 | nM | 4.42 |
| CHEMBL1701224 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1445488 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1993612 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1439815 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL2001743 | — | IC50 | > | 99000.0 | nM | - |