Assay Detail
Functional
CHEMBL1614307
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based/Microorganism Dose Confirmation HTS to Identify Inhibitors of Trypanosoma cruzi Replication. (Class of assay: confirmatory) [Related pubchem assays: 1885, 1968 ]
4060
Total Activities
4058
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 4060 | 5.98 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1506757 | — | — | 1 | 7.00 |
| CHEMBL1309132 | — | — | 1 | 7.00 |
| CHEMBL1489815 | — | — | 1 | 7.00 |
| CHEMBL1333527 | — | — | 1 | 7.00 |
| CHEMBL1588531 | — | — | 1 | 7.00 |
| CHEMBL1579600 | — | — | 1 | 7.00 |
| CHEMBL1454356 | — | — | 1 | 7.00 |
| CHEMBL64391 | ITRACONAZOLE | 4.0 | 1 | 7.00 |
| CHEMBL1315993 | — | — | 1 | 7.00 |
| CHEMBL1490099 | — | — | 1 | 6.99 |
| CHEMBL607140 | — | — | 1 | 6.99 |
| CHEMBL1375788 | — | — | 1 | 6.99 |
| CHEMBL1993291 | — | — | 1 | 6.99 |
| CHEMBL1589770 | — | — | 1 | 6.99 |
| CHEMBL1470506 | — | — | 1 | 6.99 |
| CHEMBL1448592 | — | — | 2 | 6.99 |
| CHEMBL1333111 | — | — | 1 | 6.99 |
| CHEMBL1602006 | — | — | 1 | 6.99 |
| CHEMBL1406312 | — | — | 1 | 6.99 |
| CHEMBL1517889 | — | — | 1 | 6.99 |
| CHEMBL1466872 | — | — | 1 | 6.99 |
| CHEMBL1299566 | — | — | 1 | 6.99 |
| CHEMBL3196728 | — | — | 1 | 6.99 |
| CHEMBL1437928 | — | — | 1 | 6.98 |
| CHEMBL1583933 | — | — | 1 | 6.98 |
| CHEMBL1607512 | — | — | 1 | 6.98 |
| CHEMBL1529005 | — | — | 1 | 6.98 |
| CHEMBL1508707 | — | — | 1 | 6.98 |
| CHEMBL1997747 | — | — | 1 | 6.98 |
| CHEMBL249987 | — | — | 1 | 6.98 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL64391 | ITRACONAZOLE | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1489815 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1579600 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1315993 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1588531 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1333527 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1309132 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1506757 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1454356 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1333111 | — | EC50 | = | 103.0 | nM | 6.99 |
| CHEMBL1993291 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL607140 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL1375788 | — | EC50 | = | 103.0 | nM | 6.99 |
| CHEMBL1406312 | — | EC50 | = | 103.0 | nM | 6.99 |
| CHEMBL1589770 | — | EC50 | = | 103.0 | nM | 6.99 |
| CHEMBL3196728 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL1602006 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL1470506 | — | EC50 | = | 103.0 | nM | 6.99 |
| CHEMBL1448592 | — | EC50 | = | 103.0 | nM | 6.99 |
| CHEMBL1517889 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL1299566 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL1490099 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL1466872 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL1454957 | — | EC50 | = | 105.0 | nM | 6.98 |
| CHEMBL1583933 | — | EC50 | = | 104.0 | nM | 6.98 |
| CHEMBL1508707 | — | EC50 | = | 105.0 | nM | 6.98 |
| CHEMBL1529005 | — | EC50 | = | 104.0 | nM | 6.98 |
| CHEMBL1437928 | — | EC50 | = | 105.0 | nM | 6.98 |
| CHEMBL1997747 | — | EC50 | = | 105.0 | nM | 6.98 |
| CHEMBL249987 | — | EC50 | = | 105.0 | nM | 6.98 |
| CHEMBL1599994 | — | EC50 | = | 104.0 | nM | 6.98 |
| CHEMBL1607512 | — | EC50 | = | 104.0 | nM | 6.98 |
| CHEMBL1599582 | — | EC50 | = | 106.0 | nM | 6.97 |
| CHEMBL1441053 | — | EC50 | = | 106.0 | nM | 6.97 |
| CHEMBL1546827 | — | EC50 | = | 108.0 | nM | 6.97 |
| CHEMBL1446462 | — | EC50 | = | 108.0 | nM | 6.97 |
| CHEMBL1472130 | — | EC50 | = | 107.0 | nM | 6.97 |
| CHEMBL2369174 | — | EC50 | = | 108.0 | nM | 6.97 |
| CHEMBL1518337 | — | EC50 | = | 106.0 | nM | 6.97 |
| CHEMBL1588034 | — | EC50 | = | 107.0 | nM | 6.97 |
| CHEMBL1323186 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL1427040 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL1519827 | — | EC50 | = | 111.0 | nM | 6.96 |
| CHEMBL1508476 | — | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL516194 | — | EC50 | = | 111.0 | nM | 6.96 |
| CHEMBL1401325 | — | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL1330830 | — | EC50 | = | 112.0 | nM | 6.95 |
| CHEMBL1610530 | — | EC50 | = | 113.0 | nM | 6.95 |
| CHEMBL1323545 | — | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL1503688 | — | EC50 | = | 114.0 | nM | 6.94 |