Assay Detail
Functional
CHEMBL1614370
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: High Throughput Screen to Identify Compounds that Suppress the Growth of Cells with a Deletion of the PTEN Tumor Suppressor - Dose Response. (Class of assay: confirmatory) [Related pubchem assays: 1045, 1004, 824, 999, 818, 827, 823 ]
1383
Total Activities
1382
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1383 | 4.97 | 7.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1339905 | — | — | 1 | 7.85 |
| CHEMBL1308313 | — | — | 1 | 7.07 |
| CHEMBL964 | DISULFIRAM | 4.0 | 1 | 7.06 |
| CHEMBL1303326 | — | — | 1 | 6.93 |
| CHEMBL1543295 | — | — | 1 | 6.93 |
| CHEMBL3190941 | — | — | 1 | 6.86 |
| CHEMBL123 | ELLIPTECINE | — | 1 | 6.75 |
| CHEMBL1574879 | — | — | 1 | 6.71 |
| CHEMBL1493442 | — | — | 1 | 6.66 |
| CHEMBL1425921 | — | — | 1 | 6.65 |
| CHEMBL1497549 | — | — | 1 | 6.63 |
| CHEMBL533602 | — | — | 1 | 6.63 |
| CHEMBL576409 | — | — | 1 | 6.60 |
| CHEMBL1542833 | — | — | 1 | 6.59 |
| CHEMBL1438881 | — | — | 1 | 6.53 |
| CHEMBL1588525 | — | — | 1 | 6.52 |
| CHEMBL588038 | — | — | 1 | 6.46 |
| CHEMBL1304623 | — | — | 1 | 6.41 |
| CHEMBL1424697 | — | — | 1 | 6.40 |
| CHEMBL2004157 | — | — | 1 | 6.38 |
| CHEMBL1349063 | — | — | 1 | 6.38 |
| CHEMBL1384253 | — | — | 1 | 6.31 |
| CHEMBL600734 | — | — | 1 | 6.27 |
| CHEMBL1360793 | — | — | 1 | 6.26 |
| CHEMBL1467655 | — | — | 1 | 6.26 |
| CHEMBL1490404 | — | — | 1 | 6.22 |
| CHEMBL1584754 | — | — | 1 | 6.19 |
| CHEMBL3193835 | — | — | 1 | 6.16 |
| CHEMBL1596681 | — | — | 1 | 6.14 |
| CHEMBL3197314 | — | — | 1 | 6.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1339905 | — | EC50 | = | 14.0 | nM | 7.85 |
| CHEMBL1308313 | — | EC50 | = | 85.0 | nM | 7.07 |
| CHEMBL964 | DISULFIRAM | EC50 | = | 87.0 | nM | 7.06 |
| CHEMBL1303326 | — | EC50 | = | 117.0 | nM | 6.93 |
| CHEMBL1543295 | — | EC50 | = | 117.0 | nM | 6.93 |
| CHEMBL3190941 | — | EC50 | = | 138.0 | nM | 6.86 |
| CHEMBL123 | ELLIPTECINE | EC50 | = | 177.0 | nM | 6.75 |
| CHEMBL1574879 | — | EC50 | = | 197.0 | nM | 6.71 |
| CHEMBL1493442 | — | EC50 | = | 219.0 | nM | 6.66 |
| CHEMBL1425921 | — | EC50 | = | 224.0 | nM | 6.65 |
| CHEMBL533602 | — | EC50 | = | 235.0 | nM | 6.63 |
| CHEMBL1497549 | — | EC50 | = | 234.0 | nM | 6.63 |
| CHEMBL576409 | — | EC50 | = | 249.0 | nM | 6.60 |
| CHEMBL1542833 | — | EC50 | = | 254.0 | nM | 6.59 |
| CHEMBL1438881 | — | EC50 | = | 295.0 | nM | 6.53 |
| CHEMBL1588525 | — | EC50 | = | 303.0 | nM | 6.52 |
| CHEMBL588038 | — | EC50 | = | 349.0 | nM | 6.46 |
| CHEMBL1304623 | — | EC50 | = | 389.0 | nM | 6.41 |
| CHEMBL1424697 | — | EC50 | = | 400.0 | nM | 6.40 |
| CHEMBL1349063 | — | EC50 | = | 412.0 | nM | 6.38 |
| CHEMBL2004157 | — | EC50 | = | 412.0 | nM | 6.38 |
| CHEMBL1384253 | — | EC50 | = | 487.0 | nM | 6.31 |
| CHEMBL600734 | — | EC50 | = | 540.0 | nM | 6.27 |
| CHEMBL1467655 | — | EC50 | = | 555.0 | nM | 6.26 |
| CHEMBL1360793 | — | EC50 | = | 552.0 | nM | 6.26 |
| CHEMBL1490404 | — | EC50 | = | 596.0 | nM | 6.22 |
| CHEMBL1584754 | — | EC50 | = | 650.0 | nM | 6.19 |
| CHEMBL3193835 | — | EC50 | = | 688.0 | nM | 6.16 |
| CHEMBL1596681 | — | EC50 | = | 728.0 | nM | 6.14 |
| CHEMBL1349146 | — | EC50 | = | 778.0 | nM | 6.11 |
| CHEMBL3197314 | — | EC50 | = | 777.0 | nM | 6.11 |
| CHEMBL1496534 | — | EC50 | = | 778.0 | nM | 6.11 |
| CHEMBL1460352 | — | EC50 | = | 800.0 | nM | 6.10 |
| CHEMBL601757 | — | EC50 | = | 821.0 | nM | 6.09 |
| CHEMBL1411210 | — | EC50 | = | 824.0 | nM | 6.08 |
| CHEMBL29711 | APHIDICOLIN | EC50 | = | 839.0 | nM | 6.08 |
| CHEMBL1415885 | — | EC50 | = | 850.0 | nM | 6.07 |
| CHEMBL1519279 | — | EC50 | = | 876.0 | nM | 6.06 |
| CHEMBL1347071 | — | EC50 | = | 868.0 | nM | 6.06 |
| CHEMBL1430068 | — | EC50 | = | 959.0 | nM | 6.02 |
| CHEMBL117966 | — | EC50 | = | 985.0 | nM | 6.01 |
| CHEMBL1452264 | — | EC50 | = | 1007.0 | nM | 6.00 |
| CHEMBL1499306 | — | EC50 | = | 1027.0 | nM | 5.99 |
| CHEMBL1541834 | — | EC50 | = | 1032.0 | nM | 5.99 |
| CHEMBL1569910 | — | EC50 | = | 1021.0 | nM | 5.99 |
| CHEMBL3198581 | — | EC50 | = | 1088.0 | nM | 5.96 |
| CHEMBL3192555 | — | EC50 | = | 1096.0 | nM | 5.96 |
| CHEMBL1472126 | — | EC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL1486387 | — | EC50 | = | 1121.0 | nM | 5.95 |
| CHEMBL1379675 | — | EC50 | = | 1122.0 | nM | 5.95 |