Assay Detail
Functional
CHEMBL1614384
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence-based cell-based dose response assay to identify inhibitors of NADPH oxidase 1 (NOX1). (Class of assay: confirmatory) [Related pubchem assays: 2532 (Dose response (NOX1 inhibitors, HEK/293 cells)), 1792 (Primary Screen (NOX1 inhibitors)), 1796 (Summary AID (NOX1 inhibitors)), 2545 (Confirmation screen (NOX1 inhibitors, HEK/293 cells)), 2539 (Counterscreen (NOX2, NOX3, NOX4 inhibitors)), 2541 (Confirmation screen (NOX1 inhibitors)), 1823 (Counterscreen (luminal))]
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 22 | 6.61 | 7.36 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1323615 | — | — | 1 | 7.36 |
| CHEMBL1567692 | — | — | 1 | 7.32 |
| CHEMBL1331532 | — | — | 1 | 7.28 |
| CHEMBL1401860 | — | — | 1 | 7.27 |
| CHEMBL1350157 | — | — | 1 | 7.08 |
| CHEMBL407734 | — | — | 1 | 6.81 |
| CHEMBL1449547 | — | — | 1 | 6.81 |
| CHEMBL1377821 | — | — | 1 | 6.75 |
| CHEMBL1330018 | — | — | 1 | 6.73 |
| CHEMBL1526463 | — | — | 1 | 6.60 |
| CHEMBL828 | PHENOTHIAZINE | 2.0 | 1 | 6.46 |
| CHEMBL1404241 | — | — | 1 | 6.45 |
| CHEMBL1331887 | — | — | 1 | 6.33 |
| CHEMBL1362864 | — | — | 1 | 6.00 |
| CHEMBL1437772 | — | — | 1 | 5.34 |
| CHEMBL1334632 | — | — | 1 | 5.18 |
| CHEMBL1515783 | — | — | 1 | - |
| CHEMBL1331821 | — | — | 1 | - |
| CHEMBL1357284 | — | — | 1 | - |
| CHEMBL1329357 | — | — | 1 | - |
| CHEMBL1408592 | — | — | 1 | - |
| CHEMBL1396515 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1323615 | — | IC50 | = | 44.0 | nM | 7.36 |
| CHEMBL1567692 | — | IC50 | = | 48.0 | nM | 7.32 |
| CHEMBL1331532 | — | IC50 | = | 53.0 | nM | 7.28 |
| CHEMBL1401860 | — | IC50 | = | 54.0 | nM | 7.27 |
| CHEMBL1350157 | — | IC50 | = | 83.0 | nM | 7.08 |
| CHEMBL407734 | — | IC50 | = | 156.0 | nM | 6.81 |
| CHEMBL1449547 | — | IC50 | = | 156.0 | nM | 6.81 |
| CHEMBL1377821 | — | IC50 | = | 176.0 | nM | 6.75 |
| CHEMBL1330018 | — | IC50 | = | 187.0 | nM | 6.73 |
| CHEMBL1526463 | — | IC50 | = | 252.0 | nM | 6.60 |
| CHEMBL828 | PHENOTHIAZINE | IC50 | = | 349.0 | nM | 6.46 |
| CHEMBL1404241 | — | IC50 | = | 354.0 | nM | 6.45 |
| CHEMBL1331887 | — | IC50 | = | 464.0 | nM | 6.33 |
| CHEMBL1362864 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1437772 | — | IC50 | = | 4570.0 | nM | 5.34 |
| CHEMBL1334632 | — | IC50 | = | 6603.0 | nM | 5.18 |
| CHEMBL1515783 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1331821 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1357284 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1329357 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1408592 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1396515 | — | IC50 | > | 20000.0 | nM | - |