Assay Detail
Functional
CHEMBL1614427
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: 14-3-3 protein interaction modulators Dose Response Confirmation. (Class of assay: confirmatory) [Related pubchem assays: 422 (Primary screen preceding this dose response confirmation assay.)]
52
Total Activities
52
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 52 | 4.91 | 6.07 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1502839 | — | — | 1 | 6.07 |
| CHEMBL1598223 | — | — | 1 | 5.50 |
| CHEMBL1385512 | — | — | 1 | 5.30 |
| CHEMBL2003304 | — | — | 1 | 5.14 |
| CHEMBL1544329 | — | — | 1 | 5.05 |
| CHEMBL2001481 | — | — | 1 | 5.01 |
| CHEMBL1332240 | — | — | 1 | 4.97 |
| CHEMBL1366915 | — | — | 1 | 4.74 |
| CHEMBL1328512 | — | — | 1 | 4.61 |
| CHEMBL1448942 | — | — | 1 | 4.59 |
| CHEMBL1589562 | — | — | 1 | 4.59 |
| CHEMBL1558400 | — | — | 1 | 4.52 |
| CHEMBL1501269 | — | — | 1 | 4.34 |
| CHEMBL1384321 | — | — | 1 | 4.30 |
| CHEMBL1367990 | — | — | 1 | - |
| CHEMBL1430492 | — | — | 1 | - |
| CHEMBL1390274 | — | — | 1 | - |
| CHEMBL1484912 | — | — | 1 | - |
| CHEMBL52 | NORDIHYDROGUAIARETIC ACID | — | 1 | - |
| CHEMBL1523317 | — | — | 1 | - |
| CHEMBL1529647 | — | — | 1 | - |
| CHEMBL1314409 | — | — | 1 | - |
| CHEMBL1583664 | — | — | 1 | - |
| CHEMBL1348066 | — | — | 1 | - |
| CHEMBL1563 | DAUNORUBICIN HYDROCHLORIDE | 4.0 | 1 | - |
| CHEMBL1575084 | — | — | 1 | - |
| CHEMBL1456172 | — | — | 1 | - |
| CHEMBL1582991 | — | — | 1 | - |
| CHEMBL1391466 | — | — | 1 | - |
| CHEMBL1526410 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1502839 | — | IC50 | = | 852.7 | nM | 6.07 |
| CHEMBL1598223 | — | IC50 | = | 3147.3 | nM | 5.50 |
| CHEMBL1385512 | — | IC50 | = | 5022.5 | nM | 5.30 |
| CHEMBL2003304 | — | IC50 | = | 7294.5 | nM | 5.14 |
| CHEMBL1544329 | — | IC50 | = | 8916.9 | nM | 5.05 |
| CHEMBL2001481 | — | IC50 | = | 9678.7 | nM | 5.01 |
| CHEMBL1332240 | — | IC50 | = | 10660.4 | nM | 4.97 |
| CHEMBL1366915 | — | IC50 | = | 18093.5 | nM | 4.74 |
| CHEMBL1328512 | — | IC50 | = | 24609.0 | nM | 4.61 |
| CHEMBL1448942 | — | IC50 | = | 25723.5 | nM | 4.59 |
| CHEMBL1589562 | — | IC50 | = | 25627.8 | nM | 4.59 |
| CHEMBL1558400 | — | IC50 | = | 29952.3 | nM | 4.52 |
| CHEMBL1501269 | — | IC50 | = | 45550.5 | nM | 4.34 |
| CHEMBL1384321 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL1569232 | — | IC50 | < | 44036.8 | nM | - |
| CHEMBL1200938 | METHYSERGIDE MALEATE | IC50 | > | 50000.0 | nM | - |
| CHEMBL359744 | DOXORUBICIN HYDROCHLORIDE | IC50 | < | 781.25 | nM | - |
| CHEMBL1438583 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1419748 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1498522 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1724937 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1595661 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1369154 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3190482 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1439609 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1376878 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3199764 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3216654 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL166209 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1453694 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1502394 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1606087 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1314409 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1526410 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1391466 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1582991 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1456172 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1575084 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1563 | DAUNORUBICIN HYDROCHLORIDE | IC50 | < | 781.25 | nM | - |
| CHEMBL1348066 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1583664 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1602413 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1529647 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1523317 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL52 | NORDIHYDROGUAIARETIC ACID | IC50 | > | 50000.0 | nM | - |
| CHEMBL1484912 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1390274 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1430492 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1367990 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3214300 | — | IC50 | > | 50000.0 | nM | - |