Assay Detail
Functional
CHEMBL1614455
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: A Counter Screen to identiry small molecule screen for inhibitors of the PhoP region in Salmonella Typhimurium. (Class of assay: confirmatory) [Related pubchem assays: 2253, 1863, 1981, 1874 ]
532
Total Activities
529
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 532 | 4.56 | 6.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5315124 | LEVOFLOXACIN | 4.0 | 1 | 6.43 |
| CHEMBL849 | TRICLOSAN | 4.0 | 1 | 6.31 |
| CHEMBL22 | TRIMETHOPRIM | 4.0 | 1 | 6.25 |
| CHEMBL1593697 | — | — | 1 | 6.24 |
| CHEMBL478120 | MARBOFLOXACIN | 2.0 | 1 | 6.21 |
| CHEMBL1430611 | — | — | 1 | 6.19 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | 4.0 | 1 | 6.17 |
| CHEMBL15511 | ENROFLOXACIN | 2.0 | 1 | 6.13 |
| CHEMBL351660 | — | — | 1 | 6.13 |
| CHEMBL251670 | (R)-GATIFLOXACIN | — | 1 | 6.11 |
| CHEMBL1551640 | — | — | 1 | 6.10 |
| CHEMBL4 | OFLOXACIN | 4.0 | 1 | 6.10 |
| CHEMBL9 | NORFLOXACIN | 4.0 | 1 | 6.06 |
| CHEMBL283849 | — | — | 1 | 6.03 |
| CHEMBL1315061 | — | — | 1 | 6.00 |
| CHEMBL31 | GATIFLOXACIN | 4.0 | 1 | 5.98 |
| CHEMBL601757 | — | — | 1 | 5.96 |
| CHEMBL104270 | TOSUFLOXACIN TOSYLATE | — | 1 | 5.95 |
| CHEMBL1200735 | MOXIFLOXACIN HYDROCHLORIDE | 4.0 | 1 | 5.90 |
| CHEMBL1594055 | — | — | 1 | 5.89 |
| CHEMBL1572266 | — | — | 1 | 5.87 |
| CHEMBL334707 | — | — | 1 | 5.79 |
| CHEMBL494760 | ORMETOPRIM | 2.0 | 1 | 5.69 |
| CHEMBL1428564 | PEFLOXACIN MESYLATE | -1.0 | 1 | 5.67 |
| CHEMBL1318861 | — | — | 1 | 5.64 |
| CHEMBL1485275 | — | — | 1 | 5.64 |
| CHEMBL529 | AZITHROMYCIN | 4.0 | 1 | 5.62 |
| CHEMBL1454910 | NITROXOLINE | 4.0 | 1 | 5.62 |
| CHEMBL428064 | — | — | 1 | 5.56 |
| CHEMBL1200567 | — | — | 1 | 5.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5315124 | LEVOFLOXACIN | IC50 | = | 370.0 | nM | 6.43 |
| CHEMBL849 | TRICLOSAN | IC50 | = | 490.0 | nM | 6.31 |
| CHEMBL22 | TRIMETHOPRIM | IC50 | = | 560.0 | nM | 6.25 |
| CHEMBL1593697 | — | IC50 | = | 580.0 | nM | 6.24 |
| CHEMBL478120 | MARBOFLOXACIN | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL1430611 | — | IC50 | = | 640.0 | nM | 6.19 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | IC50 | = | 670.0 | nM | 6.17 |
| CHEMBL15511 | ENROFLOXACIN | IC50 | = | 740.0 | nM | 6.13 |
| CHEMBL351660 | — | IC50 | = | 740.0 | nM | 6.13 |
| CHEMBL251670 | (R)-GATIFLOXACIN | IC50 | = | 780.0 | nM | 6.11 |
| CHEMBL1551640 | — | IC50 | = | 790.0 | nM | 6.10 |
| CHEMBL4 | OFLOXACIN | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL9 | NORFLOXACIN | IC50 | = | 880.0 | nM | 6.06 |
| CHEMBL283849 | — | IC50 | = | 930.0 | nM | 6.03 |
| CHEMBL1315061 | — | IC50 | = | 1010.0 | nM | 6.00 |
| CHEMBL31 | GATIFLOXACIN | IC50 | = | 1050.0 | nM | 5.98 |
| CHEMBL601757 | — | IC50 | = | 1090.0 | nM | 5.96 |
| CHEMBL104270 | TOSUFLOXACIN TOSYLATE | IC50 | = | 1130.0 | nM | 5.95 |
| CHEMBL1200735 | MOXIFLOXACIN HYDROCHLORIDE | IC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL1594055 | — | IC50 | = | 1280.0 | nM | 5.89 |
| CHEMBL1572266 | — | IC50 | = | 1340.0 | nM | 5.87 |
| CHEMBL334707 | — | IC50 | = | 1620.0 | nM | 5.79 |
| CHEMBL494760 | ORMETOPRIM | IC50 | = | 2030.0 | nM | 5.69 |
| CHEMBL1428564 | PEFLOXACIN MESYLATE | IC50 | = | 2150.0 | nM | 5.67 |
| CHEMBL1485275 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL1318861 | — | IC50 | = | 2280.0 | nM | 5.64 |
| CHEMBL529 | AZITHROMYCIN | IC50 | = | 2370.0 | nM | 5.62 |
| CHEMBL1454910 | NITROXOLINE | IC50 | = | 2370.0 | nM | 5.62 |
| CHEMBL428064 | — | IC50 | = | 2730.0 | nM | 5.56 |
| CHEMBL1200567 | — | IC50 | = | 2870.0 | nM | 5.54 |
| CHEMBL1604283 | — | IC50 | = | 3440.0 | nM | 5.46 |
| CHEMBL1513204 | — | IC50 | = | 3630.0 | nM | 5.44 |
| CHEMBL1545940 | — | IC50 | = | 3970.0 | nM | 5.40 |
| CHEMBL1385808 | — | IC50 | = | 4760.0 | nM | 5.32 |
| CHEMBL140425 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL1487183 | ALEXIDINE HYDROCHLORIDE | IC50 | = | 5510.0 | nM | 5.26 |
| CHEMBL1330113 | — | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL1325945 | — | IC50 | = | 5570.0 | nM | 5.25 |
| CHEMBL1333537 | — | IC50 | = | 6510.0 | nM | 5.19 |
| CHEMBL374478 | RIFAMPIN | IC50 | = | 6410.0 | nM | 5.19 |
| CHEMBL1503359 | — | IC50 | = | 6670.0 | nM | 5.18 |
| CHEMBL1579686 | — | IC50 | = | 7930.0 | nM | 5.10 |
| CHEMBL1462938 | — | IC50 | = | 8110.0 | nM | 5.09 |
| CHEMBL295619 | RUFLOXACIN | IC50 | = | 8060.0 | nM | 5.09 |
| CHEMBL1487639 | — | IC50 | = | 8120.0 | nM | 5.09 |
| CHEMBL1385206 | — | IC50 | = | 8090.0 | nM | 5.09 |
| CHEMBL497 | CLIOQUINOL | IC50 | = | 8560.0 | nM | 5.07 |
| CHEMBL139935 | — | IC50 | = | 9050.0 | nM | 5.04 |
| CHEMBL1330113 | — | IC50 | = | 9190.0 | nM | 5.04 |
| CHEMBL3189342 | — | IC50 | = | 9030.0 | nM | 5.04 |