Assay Detail
Functional
CHEMBL1738246
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: MOA HePTP Fluorescent secondary assay for identification of redox-state modulating compounds. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1059, AID1077, AID2085, AID2134, AID435032, AID521]
128
Total Activities
124
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 7 (CHEMBL2219) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 128 | 5.83 | 7.84 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1605172 | — | — | 1 | 7.84 |
| CHEMBL1322542 | — | — | 1 | 7.60 |
| CHEMBL1408579 | — | — | 1 | 7.46 |
| CHEMBL1304193 | — | — | 1 | 7.23 |
| CHEMBL1460470 | — | — | 1 | 7.18 |
| CHEMBL1608642 | — | — | 2 | 7.07 |
| CHEMBL1445488 | — | — | 1 | 6.98 |
| CHEMBL1505246 | — | — | 1 | 6.97 |
| CHEMBL1603381 | — | — | 1 | 6.90 |
| CHEMBL1407203 | — | — | 1 | 6.89 |
| CHEMBL1371869 | — | — | 1 | 6.80 |
| CHEMBL1448629 | — | — | 1 | 6.75 |
| CHEMBL1447397 | — | — | 1 | 6.71 |
| CHEMBL1501132 | — | — | 1 | 6.70 |
| CHEMBL1536896 | — | — | 1 | 6.68 |
| CHEMBL1393151 | — | — | 1 | 6.64 |
| CHEMBL1407368 | — | — | 1 | 6.59 |
| CHEMBL1449836 | — | — | 1 | 6.55 |
| CHEMBL1526088 | — | — | 1 | 6.55 |
| CHEMBL1371777 | — | — | 1 | 6.48 |
| CHEMBL1732016 | — | — | 1 | 6.43 |
| CHEMBL1414679 | — | — | 1 | 6.41 |
| CHEMBL1702580 | — | — | 1 | 6.34 |
| CHEMBL1725599 | — | — | 1 | 6.33 |
| CHEMBL1411862 | — | — | 1 | 6.32 |
| CHEMBL1424189 | — | — | 1 | 6.28 |
| CHEMBL1374242 | — | — | 2 | 6.27 |
| CHEMBL1609429 | — | — | 1 | 6.27 |
| CHEMBL1730460 | — | — | 1 | 6.26 |
| CHEMBL1372387 | — | — | 1 | 6.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1605172 | — | IC50 | = | 14.4 | nM | 7.84 |
| CHEMBL1322542 | — | IC50 | = | 25.0 | nM | 7.60 |
| CHEMBL1408579 | — | IC50 | = | 34.5 | nM | 7.46 |
| CHEMBL1304193 | — | IC50 | = | 58.6 | nM | 7.23 |
| CHEMBL1460470 | — | IC50 | = | 66.0 | nM | 7.18 |
| CHEMBL1608642 | — | IC50 | = | 84.6 | nM | 7.07 |
| CHEMBL1445488 | — | IC50 | = | 105.0 | nM | 6.98 |
| CHEMBL1505246 | — | IC50 | = | 108.0 | nM | 6.97 |
| CHEMBL1603381 | — | IC50 | = | 127.0 | nM | 6.90 |
| CHEMBL1407203 | — | IC50 | = | 129.0 | nM | 6.89 |
| CHEMBL1371869 | — | IC50 | = | 159.0 | nM | 6.80 |
| CHEMBL1448629 | — | IC50 | = | 180.0 | nM | 6.75 |
| CHEMBL1447397 | — | IC50 | = | 196.0 | nM | 6.71 |
| CHEMBL1501132 | — | IC50 | = | 198.0 | nM | 6.70 |
| CHEMBL1536896 | — | IC50 | = | 209.0 | nM | 6.68 |
| CHEMBL1393151 | — | IC50 | = | 227.0 | nM | 6.64 |
| CHEMBL1407368 | — | IC50 | = | 256.0 | nM | 6.59 |
| CHEMBL1526088 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL1449836 | — | IC50 | = | 284.0 | nM | 6.55 |
| CHEMBL1371777 | — | IC50 | = | 329.0 | nM | 6.48 |
| CHEMBL1732016 | — | IC50 | = | 373.0 | nM | 6.43 |
| CHEMBL1414679 | — | IC50 | = | 391.0 | nM | 6.41 |
| CHEMBL1702580 | — | IC50 | = | 452.0 | nM | 6.34 |
| CHEMBL1725599 | — | IC50 | = | 472.0 | nM | 6.33 |
| CHEMBL1411862 | — | IC50 | = | 476.0 | nM | 6.32 |
| CHEMBL1424189 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL1374242 | — | IC50 | = | 537.0 | nM | 6.27 |
| CHEMBL1609429 | — | IC50 | = | 537.0 | nM | 6.27 |
| CHEMBL1730460 | — | IC50 | = | 550.0 | nM | 6.26 |
| CHEMBL1735214 | — | IC50 | = | 575.0 | nM | 6.24 |
| CHEMBL1372387 | — | IC50 | = | 576.0 | nM | 6.24 |
| CHEMBL1569076 | — | IC50 | = | 588.0 | nM | 6.23 |
| CHEMBL1702303 | — | IC50 | = | 665.0 | nM | 6.18 |
| CHEMBL1714241 | — | IC50 | = | 683.0 | nM | 6.17 |
| CHEMBL1707169 | — | IC50 | = | 693.0 | nM | 6.16 |
| CHEMBL1727475 | — | IC50 | = | 766.0 | nM | 6.12 |
| CHEMBL1713063 | — | IC50 | = | 816.0 | nM | 6.09 |
| CHEMBL1500600 | — | IC50 | = | 805.0 | nM | 6.09 |
| CHEMBL1608654 | — | IC50 | = | 805.0 | nM | 6.09 |
| CHEMBL1373210 | — | IC50 | = | 819.0 | nM | 6.09 |
| CHEMBL1333996 | — | IC50 | = | 840.0 | nM | 6.08 |
| CHEMBL1374242 | — | IC50 | = | 841.0 | nM | 6.08 |
| CHEMBL1729151 | — | IC50 | = | 949.0 | nM | 6.02 |
| CHEMBL1709111 | — | IC50 | = | 1010.0 | nM | 6.00 |
| CHEMBL1500600 | — | IC50 | = | 998.0 | nM | 6.00 |
| CHEMBL1566165 | — | IC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL1448985 | — | IC50 | = | 1050.0 | nM | 5.98 |
| CHEMBL1449334 | — | IC50 | = | 1040.0 | nM | 5.98 |
| CHEMBL601167 | — | IC50 | = | 1070.0 | nM | 5.97 |
| CHEMBL1721671 | — | IC50 | = | 1090.0 | nM | 5.96 |