Assay Detail
Functional
CHEMBL1738249
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response confirmation of small molecule activators of the adaptive arm of the Unfolded Protein response via a luminescent-based reporter assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID463104, AID463126]
631
Total Activities
631
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 631 | 4.61 | 5.61 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1556884 | — | — | 1 | 5.61 |
| CHEMBL2369184 | — | — | 1 | 5.39 |
| CHEMBL1580073 | — | — | 1 | 5.37 |
| CHEMBL1377964 | — | — | 1 | 5.37 |
| CHEMBL1348169 | — | — | 1 | 5.33 |
| CHEMBL1441619 | — | — | 1 | 5.31 |
| CHEMBL3210329 | — | — | 1 | 5.27 |
| CHEMBL1539808 | — | — | 1 | 5.23 |
| CHEMBL1422301 | — | — | 1 | 5.18 |
| CHEMBL1720448 | — | — | 1 | 5.18 |
| CHEMBL1580848 | — | — | 1 | 5.11 |
| CHEMBL3193435 | — | — | 1 | 5.08 |
| CHEMBL1580664 | — | — | 1 | 5.08 |
| CHEMBL3197092 | — | — | 1 | 5.06 |
| CHEMBL1576754 | — | — | 1 | 5.05 |
| CHEMBL1535134 | — | — | 1 | 5.04 |
| CHEMBL1503152 | — | — | 1 | 5.04 |
| CHEMBL1377849 | — | — | 1 | 5.03 |
| CHEMBL1332050 | — | — | 1 | 5.01 |
| CHEMBL1517763 | — | — | 1 | 5.01 |
| CHEMBL1309018 | — | — | 1 | 5.01 |
| CHEMBL3208631 | — | — | 1 | 5.00 |
| CHEMBL1518054 | — | — | 1 | 5.00 |
| CHEMBL1981677 | — | — | 1 | 4.99 |
| CHEMBL1330510 | — | — | 1 | 4.98 |
| CHEMBL1556958 | STROBOPININ | — | 1 | 4.97 |
| CHEMBL1525745 | — | — | 1 | 4.97 |
| CHEMBL1709333 | — | — | 1 | 4.96 |
| CHEMBL1428012 | — | — | 1 | 4.96 |
| CHEMBL2007390 | — | — | 1 | 4.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1556884 | — | EC50 | = | 2460.0 | nM | 5.61 |
| CHEMBL2369184 | — | EC50 | = | 4060.0 | nM | 5.39 |
| CHEMBL1377964 | — | EC50 | = | 4310.0 | nM | 5.37 |
| CHEMBL1580073 | — | EC50 | = | 4240.0 | nM | 5.37 |
| CHEMBL1348169 | — | EC50 | = | 4670.0 | nM | 5.33 |
| CHEMBL1441619 | — | EC50 | = | 4880.0 | nM | 5.31 |
| CHEMBL3210329 | — | EC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL1539808 | — | EC50 | = | 5910.0 | nM | 5.23 |
| CHEMBL1720448 | — | EC50 | = | 6600.0 | nM | 5.18 |
| CHEMBL1422301 | — | EC50 | = | 6530.0 | nM | 5.18 |
| CHEMBL1580848 | — | EC50 | = | 7770.0 | nM | 5.11 |
| CHEMBL3193435 | — | EC50 | = | 8240.0 | nM | 5.08 |
| CHEMBL1580664 | — | EC50 | = | 8270.0 | nM | 5.08 |
| CHEMBL3197092 | — | EC50 | = | 8690.0 | nM | 5.06 |
| CHEMBL1576754 | — | EC50 | = | 8940.0 | nM | 5.05 |
| CHEMBL1503152 | — | EC50 | = | 9170.0 | nM | 5.04 |
| CHEMBL1535134 | — | EC50 | = | 9170.0 | nM | 5.04 |
| CHEMBL1377849 | — | EC50 | = | 9380.0 | nM | 5.03 |
| CHEMBL1517763 | — | EC50 | = | 9840.0 | nM | 5.01 |
| CHEMBL1332050 | — | EC50 | = | 9680.0 | nM | 5.01 |
| CHEMBL1309018 | — | EC50 | = | 9690.0 | nM | 5.01 |
| CHEMBL1518054 | — | EC50 | = | 10100.0 | nM | 5.00 |
| CHEMBL3208631 | — | EC50 | = | 10100.0 | nM | 5.00 |
| CHEMBL1981677 | — | EC50 | = | 10300.0 | nM | 4.99 |
| CHEMBL1330510 | — | EC50 | = | 10400.0 | nM | 4.98 |
| CHEMBL1525745 | — | EC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL1556958 | STROBOPININ | EC50 | = | 10800.0 | nM | 4.97 |
| CHEMBL2007390 | — | EC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL1428012 | — | EC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL1709333 | — | EC50 | = | 11100.0 | nM | 4.96 |
| CHEMBL3208014 | — | EC50 | = | 11600.0 | nM | 4.94 |
| CHEMBL1485665 | — | EC50 | = | 11700.0 | nM | 4.93 |
| CHEMBL1986073 | — | EC50 | = | 11800.0 | nM | 4.93 |
| CHEMBL1303719 | — | EC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL1508334 | — | EC50 | = | 11900.0 | nM | 4.92 |
| CHEMBL1544133 | — | EC50 | = | 11900.0 | nM | 4.92 |
| CHEMBL1383793 | — | EC50 | = | 12100.0 | nM | 4.92 |
| CHEMBL3193533 | — | EC50 | = | 12200.0 | nM | 4.91 |
| CHEMBL1392765 | — | EC50 | = | 13200.0 | nM | 4.88 |
| CHEMBL1341399 | — | EC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL1716112 | — | EC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL3209920 | — | EC50 | = | 13500.0 | nM | 4.87 |
| CHEMBL1724535 | — | EC50 | = | 13700.0 | nM | 4.86 |
| CHEMBL1496189 | — | EC50 | = | 14600.0 | nM | 4.84 |
| CHEMBL1351044 | — | EC50 | = | 15100.0 | nM | 4.82 |
| CHEMBL2000338 | — | EC50 | = | 15300.0 | nM | 4.82 |
| CHEMBL1593896 | — | EC50 | = | 15300.0 | nM | 4.82 |
| CHEMBL1722190 | — | EC50 | = | 15200.0 | nM | 4.82 |
| CHEMBL1324256 | — | EC50 | = | 15600.0 | nM | 4.81 |
| CHEMBL1500686 | — | EC50 | = | 15500.0 | nM | 4.81 |