Assay Detail
Functional
CHEMBL1738494
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response cytotoxicity of uHTS chemical inhibitors of T-cell specific antigen receptor-induced NF-kB activation in a HEK-293T cell line using a luminescence assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID435003, AID435012, AID489041]
694
Total Activities
693
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | HEK-293T |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 694 | 4.45 | 6.36 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3189714 | — | — | 1 | 6.36 |
| CHEMBL3195749 | — | — | 1 | 6.01 |
| CHEMBL1593286 | — | — | 1 | 5.80 |
| CHEMBL578512 | — | — | 1 | 5.70 |
| CHEMBL1467999 | — | — | 1 | 5.63 |
| CHEMBL1452795 | — | — | 1 | 5.50 |
| CHEMBL1418818 | — | — | 1 | 5.43 |
| CHEMBL1987894 | — | — | 1 | 5.40 |
| CHEMBL578502 | — | — | 1 | 5.39 |
| CHEMBL3191855 | — | — | 1 | 5.38 |
| CHEMBL1463659 | — | — | 1 | 5.37 |
| CHEMBL579318 | — | — | 1 | 5.12 |
| CHEMBL601757 | — | — | 1 | 5.03 |
| CHEMBL1564737 | — | — | 1 | 4.99 |
| CHEMBL1571885 | — | — | 1 | 4.77 |
| CHEMBL1409606 | — | — | 1 | 4.76 |
| CHEMBL1971727 | — | — | 1 | 4.74 |
| CHEMBL1716112 | — | — | 1 | 4.73 |
| CHEMBL1331593 | — | — | 1 | 4.71 |
| CHEMBL1335846 | — | — | 1 | 4.69 |
| CHEMBL1538246 | — | — | 1 | 4.68 |
| CHEMBL1339245 | — | — | 1 | 4.67 |
| CHEMBL1497812 | — | — | 1 | 4.65 |
| CHEMBL1491847 | — | — | 1 | 4.64 |
| CHEMBL1382884 | — | — | 1 | 4.61 |
| CHEMBL1382438 | — | — | 1 | 4.60 |
| CHEMBL1396209 | — | — | 1 | 4.59 |
| CHEMBL1448642 | — | — | 1 | 4.57 |
| CHEMBL1401272 | — | — | 1 | 4.56 |
| CHEMBL1978733 | — | — | 1 | 4.55 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3189714 | — | IC50 | = | 440.0 | nM | 6.36 |
| CHEMBL3195749 | — | IC50 | = | 980.0 | nM | 6.01 |
| CHEMBL1593286 | — | IC50 | = | 1580.0 | nM | 5.80 |
| CHEMBL578512 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL1467999 | — | IC50 | = | 2350.0 | nM | 5.63 |
| CHEMBL1452795 | — | IC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL1418818 | — | IC50 | = | 3730.0 | nM | 5.43 |
| CHEMBL1987894 | — | IC50 | = | 3960.0 | nM | 5.40 |
| CHEMBL578502 | — | IC50 | = | 4030.0 | nM | 5.39 |
| CHEMBL3191855 | — | IC50 | = | 4190.0 | nM | 5.38 |
| CHEMBL1463659 | — | IC50 | = | 4260.0 | nM | 5.37 |
| CHEMBL579318 | — | IC50 | = | 7670.0 | nM | 5.12 |
| CHEMBL601757 | — | IC50 | = | 9410.0 | nM | 5.03 |
| CHEMBL1564737 | — | IC50 | = | 10200.0 | nM | 4.99 |
| CHEMBL1571885 | — | IC50 | = | 16900.0 | nM | 4.77 |
| CHEMBL1409606 | — | IC50 | = | 17300.0 | nM | 4.76 |
| CHEMBL1971727 | — | IC50 | = | 18100.0 | nM | 4.74 |
| CHEMBL1716112 | — | IC50 | = | 18600.0 | nM | 4.73 |
| CHEMBL1331593 | — | IC50 | = | 19500.0 | nM | 4.71 |
| CHEMBL1335846 | — | IC50 | = | 20300.0 | nM | 4.69 |
| CHEMBL1538246 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL1339245 | — | IC50 | = | 21500.0 | nM | 4.67 |
| CHEMBL1497812 | — | IC50 | = | 22400.0 | nM | 4.65 |
| CHEMBL1491847 | — | IC50 | = | 22800.0 | nM | 4.64 |
| CHEMBL1382884 | — | IC50 | = | 24800.0 | nM | 4.61 |
| CHEMBL1382438 | — | IC50 | = | 25300.0 | nM | 4.60 |
| CHEMBL1396209 | — | IC50 | = | 25900.0 | nM | 4.59 |
| CHEMBL1448642 | — | IC50 | = | 27200.0 | nM | 4.57 |
| CHEMBL1401272 | — | IC50 | = | 27800.0 | nM | 4.56 |
| CHEMBL551783 | — | IC50 | = | 28300.0 | nM | 4.55 |
| CHEMBL1978733 | — | IC50 | = | 28100.0 | nM | 4.55 |
| CHEMBL1432251 | — | IC50 | = | 27900.0 | nM | 4.55 |
| CHEMBL1514534 | — | IC50 | = | 28500.0 | nM | 4.54 |
| CHEMBL1481849 | — | IC50 | = | 29000.0 | nM | 4.54 |
| CHEMBL1344225 | — | IC50 | = | 29800.0 | nM | 4.53 |
| CHEMBL1407659 | — | IC50 | = | 29600.0 | nM | 4.53 |
| CHEMBL1377737 | — | IC50 | = | 31500.0 | nM | 4.50 |
| CHEMBL1357385 | — | IC50 | = | 32500.0 | nM | 4.49 |
| CHEMBL1574879 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL576409 | — | IC50 | = | 33100.0 | nM | 4.48 |
| CHEMBL1606309 | — | IC50 | = | 33400.0 | nM | 4.48 |
| CHEMBL1491324 | — | IC50 | = | 34300.0 | nM | 4.46 |
| CHEMBL562566 | — | IC50 | = | 35900.0 | nM | 4.45 |
| CHEMBL1374527 | — | IC50 | = | 36500.0 | nM | 4.44 |
| CHEMBL1304363 | — | IC50 | = | 36800.0 | nM | 4.43 |
| CHEMBL1417019 | MITOXANTRONE HYDROCHLORIDE | IC50 | = | 37900.0 | nM | 4.42 |
| CHEMBL1537481 | — | IC50 | = | 38100.0 | nM | 4.42 |
| CHEMBL1344838 | — | IC50 | = | 38000.0 | nM | 4.42 |
| CHEMBL1481347 | — | IC50 | = | 38400.0 | nM | 4.42 |
| CHEMBL1448627 | — | IC50 | = | 39800.0 | nM | 4.40 |