Assay Detail
Functional
CHEMBL1738502
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 6 (SENP6) using a Luminescent assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2575, AID2582, AID2599]
704
Total Activities
704
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 704 | 4.95 | 6.73 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3196451 | — | — | 1 | 6.73 |
| CHEMBL1402456 | — | — | 1 | 6.46 |
| CHEMBL1449923 | — | — | 1 | 6.22 |
| CHEMBL1998302 | — | — | 1 | 6.13 |
| CHEMBL1417815 | — | — | 1 | 6.10 |
| CHEMBL281980 | — | — | 1 | 6.10 |
| CHEMBL1506796 | — | — | 1 | 6.10 |
| CHEMBL1969046 | — | — | 1 | 6.09 |
| CHEMBL205040 | — | — | 1 | 6.09 |
| CHEMBL1477061 | — | — | 1 | 6.08 |
| CHEMBL3191962 | — | — | 1 | 6.07 |
| CHEMBL1471498 | — | — | 1 | 6.03 |
| CHEMBL1421255 | — | — | 1 | 6.02 |
| CHEMBL1376622 | — | — | 1 | 6.01 |
| CHEMBL1575869 | — | — | 1 | 6.01 |
| CHEMBL1475128 | — | — | 1 | 5.97 |
| CHEMBL1542328 | — | — | 1 | 5.96 |
| CHEMBL1967857 | — | — | 1 | 5.94 |
| CHEMBL1418096 | — | — | 1 | 5.90 |
| CHEMBL3195102 | — | — | 1 | 5.88 |
| CHEMBL1988780 | — | — | 1 | 5.85 |
| CHEMBL1584379 | — | — | 1 | 5.85 |
| CHEMBL595840 | — | — | 1 | 5.82 |
| CHEMBL1438722 | — | — | 1 | 5.78 |
| CHEMBL3197982 | — | — | 1 | 5.76 |
| CHEMBL1379448 | — | — | 1 | 5.74 |
| CHEMBL3195749 | — | — | 1 | 5.73 |
| CHEMBL36536 | — | — | 1 | 5.73 |
| CHEMBL1421377 | — | — | 1 | 5.72 |
| CHEMBL2000196 | — | — | 1 | 5.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3196451 | — | IC50 | = | 186.0 | nM | 6.73 |
| CHEMBL1402456 | — | IC50 | = | 345.0 | nM | 6.46 |
| CHEMBL1449923 | — | IC50 | = | 596.0 | nM | 6.22 |
| CHEMBL1998302 | — | IC50 | = | 743.0 | nM | 6.13 |
| CHEMBL1417815 | — | IC50 | = | 802.0 | nM | 6.10 |
| CHEMBL281980 | — | IC50 | = | 789.0 | nM | 6.10 |
| CHEMBL1506796 | — | IC50 | = | 787.0 | nM | 6.10 |
| CHEMBL1969046 | — | IC50 | = | 819.0 | nM | 6.09 |
| CHEMBL205040 | — | IC50 | = | 805.0 | nM | 6.09 |
| CHEMBL1477061 | — | IC50 | = | 838.0 | nM | 6.08 |
| CHEMBL3191962 | — | IC50 | = | 849.0 | nM | 6.07 |
| CHEMBL1471498 | — | IC50 | = | 936.0 | nM | 6.03 |
| CHEMBL1421255 | — | IC50 | = | 961.0 | nM | 6.02 |
| CHEMBL1376622 | — | IC50 | = | 984.0 | nM | 6.01 |
| CHEMBL1575869 | — | IC50 | = | 986.0 | nM | 6.01 |
| CHEMBL1475128 | — | IC50 | = | 1080.0 | nM | 5.97 |
| CHEMBL1542328 | — | IC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL1967857 | — | IC50 | = | 1150.0 | nM | 5.94 |
| CHEMBL1418096 | — | IC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL3195102 | — | IC50 | = | 1310.0 | nM | 5.88 |
| CHEMBL1988780 | — | IC50 | = | 1420.0 | nM | 5.85 |
| CHEMBL1584379 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL595840 | — | IC50 | = | 1510.0 | nM | 5.82 |
| CHEMBL1438722 | — | IC50 | = | 1650.0 | nM | 5.78 |
| CHEMBL3197982 | — | IC50 | = | 1720.0 | nM | 5.76 |
| CHEMBL1379448 | — | IC50 | = | 1810.0 | nM | 5.74 |
| CHEMBL3195749 | — | IC50 | = | 1860.0 | nM | 5.73 |
| CHEMBL36536 | — | IC50 | = | 1860.0 | nM | 5.73 |
| CHEMBL1421377 | — | IC50 | = | 1890.0 | nM | 5.72 |
| CHEMBL2000196 | — | IC50 | = | 1910.0 | nM | 5.72 |
| CHEMBL1307406 | — | IC50 | = | 2010.0 | nM | 5.70 |
| CHEMBL3194086 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL1415156 | — | IC50 | = | 2030.0 | nM | 5.69 |
| CHEMBL1380580 | — | IC50 | = | 2030.0 | nM | 5.69 |
| CHEMBL3209654 | — | IC50 | = | 2090.0 | nM | 5.68 |
| CHEMBL1469807 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL3191218 | — | IC50 | = | 2160.0 | nM | 5.67 |
| CHEMBL1497070 | — | IC50 | = | 2210.0 | nM | 5.66 |
| CHEMBL1576896 | — | IC50 | = | 2210.0 | nM | 5.66 |
| CHEMBL1544489 | — | IC50 | = | 2190.0 | nM | 5.66 |
| CHEMBL1624350 | — | IC50 | = | 2240.0 | nM | 5.65 |
| CHEMBL1409039 | — | IC50 | = | 2250.0 | nM | 5.65 |
| CHEMBL1392911 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL1349748 | — | IC50 | = | 2360.0 | nM | 5.63 |
| CHEMBL3198635 | — | IC50 | = | 2340.0 | nM | 5.63 |
| CHEMBL1535503 | — | IC50 | = | 2390.0 | nM | 5.62 |
| CHEMBL1450897 | — | IC50 | = | 2370.0 | nM | 5.62 |
| CHEMBL1521051 | — | IC50 | = | 2370.0 | nM | 5.62 |
| CHEMBL1501990 | — | IC50 | = | 2390.0 | nM | 5.62 |
| CHEMBL1534289 | — | IC50 | = | 2380.0 | nM | 5.62 |