Assay Detail
Functional
CHEMBL1738579
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of inhibitors of hexokinase domain containing I (HKDC1). (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493160, AID493190]
215
Total Activities
215
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 215 | 5.02 | 5.99 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1454614 | — | — | 1 | 5.99 |
| CHEMBL1395907 | — | — | 1 | 5.87 |
| CHEMBL1728280 | — | — | 1 | 5.81 |
| CHEMBL1362935 | — | — | 1 | 5.79 |
| CHEMBL3199539 | — | — | 1 | 5.78 |
| CHEMBL1968732 | — | — | 1 | 5.75 |
| CHEMBL27953 | — | — | 1 | 5.66 |
| CHEMBL1724454 | — | — | 1 | 5.65 |
| CHEMBL1368625 | — | — | 1 | 5.64 |
| CHEMBL1310221 | — | — | 1 | 5.63 |
| CHEMBL1721095 | — | — | 1 | 5.61 |
| CHEMBL592124 | — | — | 1 | 5.61 |
| CHEMBL1451931 | — | — | 1 | 5.60 |
| CHEMBL448515 | 2,6-DIMETHOXYQUINONE | — | 1 | 5.60 |
| CHEMBL1999630 | — | — | 1 | 5.60 |
| CHEMBL1706640 | — | — | 1 | 5.59 |
| CHEMBL1329141 | — | — | 1 | 5.59 |
| CHEMBL1964361 | — | — | 1 | 5.57 |
| CHEMBL1366206 | — | — | 1 | 5.57 |
| CHEMBL1998302 | — | — | 1 | 5.56 |
| CHEMBL1721986 | — | — | 1 | 5.54 |
| CHEMBL1342410 | — | — | 1 | 5.53 |
| CHEMBL2003651 | — | — | 1 | 5.52 |
| CHEMBL1717890 | — | — | 1 | 5.51 |
| CHEMBL429095 | — | — | 1 | 5.50 |
| CHEMBL1347253 | — | — | 1 | 5.50 |
| CHEMBL1567670 | — | — | 1 | 5.50 |
| CHEMBL1729300 | — | — | 1 | 5.48 |
| CHEMBL1359359 | — | — | 1 | 5.47 |
| CHEMBL1710429 | — | — | 1 | 5.47 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1454614 | — | IC50 | = | 1020.0 | nM | 5.99 |
| CHEMBL1395907 | — | IC50 | = | 1340.0 | nM | 5.87 |
| CHEMBL1728280 | — | IC50 | = | 1560.0 | nM | 5.81 |
| CHEMBL1362935 | — | IC50 | = | 1610.0 | nM | 5.79 |
| CHEMBL3199539 | — | IC50 | = | 1680.0 | nM | 5.78 |
| CHEMBL1968732 | — | IC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL27953 | — | IC50 | = | 2180.0 | nM | 5.66 |
| CHEMBL1724454 | — | IC50 | = | 2230.0 | nM | 5.65 |
| CHEMBL1368625 | — | IC50 | = | 2310.0 | nM | 5.64 |
| CHEMBL1310221 | — | IC50 | = | 2320.0 | nM | 5.63 |
| CHEMBL592124 | — | IC50 | = | 2460.0 | nM | 5.61 |
| CHEMBL1721095 | — | IC50 | = | 2470.0 | nM | 5.61 |
| CHEMBL1999630 | — | IC50 | = | 2530.0 | nM | 5.60 |
| CHEMBL1451931 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL448515 | 2,6-DIMETHOXYQUINONE | IC50 | = | 2490.0 | nM | 5.60 |
| CHEMBL1329141 | — | IC50 | = | 2570.0 | nM | 5.59 |
| CHEMBL1706640 | — | IC50 | = | 2560.0 | nM | 5.59 |
| CHEMBL1964361 | — | IC50 | = | 2690.0 | nM | 5.57 |
| CHEMBL1366206 | — | IC50 | = | 2720.0 | nM | 5.57 |
| CHEMBL1998302 | — | IC50 | = | 2740.0 | nM | 5.56 |
| CHEMBL1721986 | — | IC50 | = | 2880.0 | nM | 5.54 |
| CHEMBL1342410 | — | IC50 | = | 2960.0 | nM | 5.53 |
| CHEMBL2003651 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL1717890 | — | IC50 | = | 3090.0 | nM | 5.51 |
| CHEMBL429095 | — | IC50 | = | 3150.0 | nM | 5.50 |
| CHEMBL1567670 | — | IC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL1347253 | — | IC50 | = | 3160.0 | nM | 5.50 |
| CHEMBL1729300 | — | IC50 | = | 3330.0 | nM | 5.48 |
| CHEMBL1301125 | — | IC50 | = | 3350.0 | nM | 5.47 |
| CHEMBL1710429 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL1345851 | — | IC50 | = | 3390.0 | nM | 5.47 |
| CHEMBL1359359 | — | IC50 | = | 3350.0 | nM | 5.47 |
| CHEMBL1376835 | — | IC50 | = | 3450.0 | nM | 5.46 |
| CHEMBL1714002 | — | IC50 | = | 3560.0 | nM | 5.45 |
| CHEMBL1996724 | — | IC50 | = | 3720.0 | nM | 5.43 |
| CHEMBL1522846 | — | IC50 | = | 3730.0 | nM | 5.43 |
| CHEMBL1540682 | — | IC50 | = | 3810.0 | nM | 5.42 |
| CHEMBL1401606 | — | IC50 | = | 3810.0 | nM | 5.42 |
| CHEMBL3197637 | — | IC50 | = | 3840.0 | nM | 5.42 |
| CHEMBL1704261 | — | IC50 | = | 3930.0 | nM | 5.41 |
| CHEMBL1356785 | — | IC50 | = | 4090.0 | nM | 5.39 |
| CHEMBL1982305 | — | IC50 | = | 4310.0 | nM | 5.37 |
| CHEMBL456881 | DEOXYVASICINONE | IC50 | = | 4320.0 | nM | 5.37 |
| CHEMBL1432707 | — | IC50 | = | 4410.0 | nM | 5.36 |
| CHEMBL1699845 | — | IC50 | = | 4470.0 | nM | 5.35 |
| CHEMBL1716550 | — | IC50 | = | 4580.0 | nM | 5.34 |
| CHEMBL1342337 | — | IC50 | = | 4720.0 | nM | 5.33 |
| CHEMBL1564699 | — | IC50 | = | 4670.0 | nM | 5.33 |
| CHEMBL1337591 | — | IC50 | = | 4710.0 | nM | 5.33 |
| CHEMBL3190880 | — | IC50 | = | 4780.0 | nM | 5.32 |