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Compound Detail

CHEMBL1359359

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CNCc1ccccc1Sc1cc(O)ccc1O.O=C(O)/C=C\C(=O)O

Basic Information

ChEMBL ID CHEMBL1359359
Phase Preclinical
Structure Type MOL
InChI Key AGYMFYABMLHWEH-BTJKTKAUSA-N
Parent Compound CHEMBL1618557
Active Moiety CHEMBL1618557
5
Targets
7
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

261.4
MW (Da)
2.97
ALogP
4
HBA
3
HBD
52.5
PSA (Ų)
0.74
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C18H19NO6S
MW 377.42
Aromatic Rings 2
Heavy Atoms 18
NP-Likeness 0.29

Activity Summary

IC50 7 meas. best 5.65

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase
CHEMBL1741212
IC50 5.65 4.955 2230.0 2
Hexokinase HKDC1
CHEMBL1741200
IC50 5.47 5.405 3350.0 2
Induced myeloid leukemia cell differentiation protein Mcl-1
CHEMBL4361
IC50 5.35 5.35 4503.7 1
C-C chemokine receptor type 6
CHEMBL4423
IC50 4.63 4.63 23500.0 1
Glucose-6-phosphate 1-dehydrogenase
CHEMBL5347
IC50 4.57 4.57 26900.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine