Assay Detail
Functional
CHEMBL1738619
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of activators of hexokinase domain containing I (HKDC1) in the hexokinase 1 selectivity assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493187, AID493207]
101
Total Activities
101
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 101 | 4.59 | 5.97 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1734083 | — | — | 1 | 5.97 |
| CHEMBL1790033 | — | — | 1 | 5.28 |
| CHEMBL1312377 | — | — | 1 | 5.18 |
| CHEMBL1576392 | — | — | 1 | 5.12 |
| CHEMBL1478479 | — | — | 1 | 5.09 |
| CHEMBL1461738 | — | — | 1 | 5.08 |
| CHEMBL1578997 | — | — | 1 | 4.97 |
| CHEMBL1704311 | — | — | 1 | 4.93 |
| CHEMBL1558692 | — | — | 1 | 4.87 |
| CHEMBL1706392 | — | — | 1 | 4.85 |
| CHEMBL1454194 | — | — | 1 | 4.82 |
| CHEMBL1482926 | — | — | 1 | 4.79 |
| CHEMBL1432378 | — | — | 1 | 4.76 |
| CHEMBL263972 | — | — | 1 | 4.75 |
| CHEMBL1589350 | — | — | 1 | 4.75 |
| CHEMBL1325587 | — | — | 1 | 4.74 |
| CHEMBL1345979 | — | — | 1 | 4.71 |
| CHEMBL1299995 | — | — | 1 | 4.70 |
| CHEMBL1434002 | — | — | 1 | 4.68 |
| CHEMBL1501771 | — | — | 1 | 4.68 |
| CHEMBL1438779 | — | — | 1 | 4.68 |
| CHEMBL1545605 | — | — | 1 | 4.66 |
| CHEMBL1419292 | — | — | 1 | 4.62 |
| CHEMBL1344977 | — | — | 1 | 4.62 |
| CHEMBL1523347 | — | — | 1 | 4.61 |
| CHEMBL1587286 | — | — | 1 | 4.54 |
| CHEMBL1371983 | — | — | 1 | 4.53 |
| CHEMBL1559226 | — | — | 1 | 4.53 |
| CHEMBL1471660 | — | — | 1 | 4.53 |
| CHEMBL1308783 | — | — | 1 | 4.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1734083 | — | EC50 | = | 1060.0 | nM | 5.97 |
| CHEMBL1790033 | — | EC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL1312377 | — | EC50 | = | 6540.0 | nM | 5.18 |
| CHEMBL1576392 | — | EC50 | = | 7650.0 | nM | 5.12 |
| CHEMBL1478479 | — | EC50 | = | 8100.0 | nM | 5.09 |
| CHEMBL1461738 | — | EC50 | = | 8260.0 | nM | 5.08 |
| CHEMBL1578997 | — | EC50 | = | 10600.0 | nM | 4.97 |
| CHEMBL1704311 | — | EC50 | = | 11800.0 | nM | 4.93 |
| CHEMBL1558692 | — | EC50 | = | 13600.0 | nM | 4.87 |
| CHEMBL1706392 | — | EC50 | = | 14200.0 | nM | 4.85 |
| CHEMBL1454194 | — | EC50 | = | 15300.0 | nM | 4.82 |
| CHEMBL1482926 | — | EC50 | = | 16300.0 | nM | 4.79 |
| CHEMBL1432378 | — | EC50 | = | 17400.0 | nM | 4.76 |
| CHEMBL1589350 | — | EC50 | = | 17800.0 | nM | 4.75 |
| CHEMBL263972 | — | EC50 | = | 17900.0 | nM | 4.75 |
| CHEMBL1325587 | — | EC50 | = | 18200.0 | nM | 4.74 |
| CHEMBL1345979 | — | EC50 | = | 19300.0 | nM | 4.71 |
| CHEMBL1299995 | — | EC50 | = | 20100.0 | nM | 4.70 |
| CHEMBL1434002 | — | EC50 | = | 21100.0 | nM | 4.68 |
| CHEMBL1501771 | — | EC50 | = | 21100.0 | nM | 4.68 |
| CHEMBL1438779 | — | EC50 | = | 20800.0 | nM | 4.68 |
| CHEMBL1545605 | — | EC50 | = | 21700.0 | nM | 4.66 |
| CHEMBL1419292 | — | EC50 | = | 23900.0 | nM | 4.62 |
| CHEMBL1344977 | — | EC50 | = | 24000.0 | nM | 4.62 |
| CHEMBL1523347 | — | EC50 | = | 24700.0 | nM | 4.61 |
| CHEMBL1587286 | — | EC50 | = | 28900.0 | nM | 4.54 |
| CHEMBL1559226 | — | EC50 | = | 29700.0 | nM | 4.53 |
| CHEMBL1471660 | — | EC50 | = | 29500.0 | nM | 4.53 |
| CHEMBL1371983 | — | EC50 | = | 29400.0 | nM | 4.53 |
| CHEMBL1308783 | — | EC50 | = | 30800.0 | nM | 4.51 |
| CHEMBL1464186 | — | EC50 | = | 32000.0 | nM | 4.50 |
| CHEMBL1546933 | — | EC50 | = | 32200.0 | nM | 4.49 |
| CHEMBL1705697 | — | EC50 | = | 34100.0 | nM | 4.47 |
| CHEMBL1527942 | — | EC50 | = | 35100.0 | nM | 4.46 |
| CHEMBL1338355 | — | EC50 | = | 34500.0 | nM | 4.46 |
| CHEMBL1382826 | — | EC50 | = | 36700.0 | nM | 4.43 |
| CHEMBL1430796 | — | EC50 | = | 37400.0 | nM | 4.43 |
| CHEMBL1498652 | — | EC50 | = | 37100.0 | nM | 4.43 |
| CHEMBL1444349 | — | EC50 | = | 37900.0 | nM | 4.42 |
| CHEMBL1582527 | — | EC50 | = | 39400.0 | nM | 4.41 |
| CHEMBL1968355 | — | EC50 | = | 39900.0 | nM | 4.40 |
| CHEMBL1318817 | — | EC50 | = | 41900.0 | nM | 4.38 |
| CHEMBL51085 | EBSELEN | EC50 | = | 41900.0 | nM | 4.38 |
| CHEMBL1417967 | — | EC50 | = | 41300.0 | nM | 4.38 |
| CHEMBL3195968 | — | EC50 | = | 42300.0 | nM | 4.37 |
| CHEMBL1432648 | — | EC50 | = | 46000.0 | nM | 4.34 |
| CHEMBL1339349 | — | EC50 | = | 46800.0 | nM | 4.33 |
| CHEMBL1604990 | — | EC50 | = | 47400.0 | nM | 4.32 |
| CHEMBL1330332 | — | EC50 | = | 49300.0 | nM | 4.31 |
| CHEMBL1708074 | — | EC50 | = | 49600.0 | nM | 4.30 |