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Compound Detail

CHEMBL1318817

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COc1cc(N=c2ssnc2Cl)c(OC)cc1Cl

Basic Information

ChEMBL ID CHEMBL1318817
Phase Preclinical
Structure Type MOL
InChI Key VOQMETKMNGYFQC-UHFFFAOYSA-N
6
Targets
8
Activities
2
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

323.2
MW (Da)
3.76
ALogP
6
HBA
0
HBD
43.7
PSA (Ų)
0.81
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C10H8Cl2N2O2S2
MW 323.23
Aromatic Rings 2
Heavy Atoms 18
NP-Likeness -1.09

Activity Summary

IC50 6 meas. best 5.05
EC50 2 meas. best 4.57

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
DNA dC->dU-editing enzyme APOBEC-3G
CHEMBL1741217
IC50 5.05 5.05 8830.0 1
Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase
CHEMBL1741212
IC50 4.87 4.6133 13500.0 3
Hexokinase HKDC1
CHEMBL1741200
EC50 4.57 4.57 27200.0 1
Hexokinase-1
CHEMBL2688
EC50 4.38 4.38 41900.0 1
Glucose-6-phosphate 1-dehydrogenase
CHEMBL5347
IC50 4.16 4.16 68800.0 1
Unchecked
CHEMBL612545
IC50 4.04 4.04 92148.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine