Assay Detail
Functional
CHEMBL1776697
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Antifibrotic activity against rat HSC-T6 cells assessed as inhibition of proliferation after 48 hrs by BrdU incorporation assay
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Cell Type | HSC-T6 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Antifibrotic constituents of Alnus firma on hepatic stellate cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 4.52 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL297453 | EPIGALOCATECHIN GALLATE | 3.0 | 1 | 5.00 |
| CHEMBL464274 | DEHYDROHIRSUTANONOL | — | 1 | 4.85 |
| CHEMBL1774776 | — | — | 1 | 4.62 |
| CHEMBL330645 | PLATYPHYLLENONE | — | 1 | 4.46 |
| CHEMBL1774771 | — | — | 1 | 4.46 |
| CHEMBL1774773 | — | — | 1 | 4.41 |
| CHEMBL464362 | — | — | 1 | 4.33 |
| CHEMBL1087992 | PLATYPHYLLONE | — | 1 | 4.26 |
| CHEMBL1774774 | — | — | 1 | 4.26 |
| CHEMBL1774721 | — | — | 1 | - |
| CHEMBL598970 | ALNUSIDE B | — | 1 | - |
| CHEMBL1774772 | — | — | 1 | - |
| CHEMBL464570 | OREGONIN | — | 1 | - |
| CHEMBL1774775 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL297453 | EPIGALOCATECHIN GALLATE | IC50 | = | 9900.0 | nM | 5.00 |
| CHEMBL464274 | DEHYDROHIRSUTANONOL | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL1774776 | — | IC50 | = | 23900.0 | nM | 4.62 |
| CHEMBL330645 | PLATYPHYLLENONE | IC50 | = | 34700.0 | nM | 4.46 |
| CHEMBL1774771 | — | IC50 | = | 34900.0 | nM | 4.46 |
| CHEMBL1774773 | — | IC50 | = | 39100.0 | nM | 4.41 |
| CHEMBL464362 | — | IC50 | = | 46200.0 | nM | 4.33 |
| CHEMBL1087992 | PLATYPHYLLONE | IC50 | = | 54900.0 | nM | 4.26 |
| CHEMBL1774774 | — | IC50 | = | 54900.0 | nM | 4.26 |
| CHEMBL1774721 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL598970 | ALNUSIDE B | IC50 | > | 100000.0 | nM | - |
| CHEMBL1774772 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL464570 | OREGONIN | IC50 | > | 100000.0 | nM | - |
| CHEMBL1774775 | — | IC50 | > | 100000.0 | nM | - |