Assay Detail
Functional
CHEMBL1794457
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Counterscreen for agonists of heterodimerization of the mu 1 (OPRM1) and delta 1 (OPRD1) opioid receptors: Luminescence-based cell-based high throughput dose response assay to identify agonists of OPRM1 homodimerization. (Class of assay: confirmatory)
229
Total Activities
228
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 229 | 4.77 | 6.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1732484 | — | — | 1 | 6.30 |
| CHEMBL1200531 | ALFENTANIL HYDROCHLORIDE | 4.0 | 1 | 6.11 |
| CHEMBL1717557 | — | — | 1 | 5.85 |
| CHEMBL1463894 | — | — | 1 | 5.62 |
| CHEMBL1307063 | — | — | 1 | 5.56 |
| CHEMBL1331866 | — | — | 1 | 5.55 |
| CHEMBL1581674 | — | — | 1 | 5.48 |
| CHEMBL1700847 | — | — | 1 | 5.44 |
| CHEMBL1380599 | — | — | 1 | 5.38 |
| CHEMBL1416425 | — | — | 1 | 5.33 |
| CHEMBL1388222 | — | — | 1 | 5.33 |
| CHEMBL1522542 | — | — | 1 | 5.32 |
| CHEMBL1609119 | — | — | 1 | 5.29 |
| CHEMBL542581 | PHENCYCLIDINE HYDROCHLORIDE | -1.0 | 1 | 5.20 |
| CHEMBL1698841 | — | — | 1 | 5.12 |
| CHEMBL1531675 | — | — | 1 | 5.00 |
| CHEMBL1426979 | — | — | 1 | 4.99 |
| CHEMBL1460676 | — | — | 1 | 4.99 |
| CHEMBL1586285 | — | — | 1 | 4.97 |
| CHEMBL1705302 | — | — | 1 | 4.96 |
| CHEMBL1720091 | — | — | 1 | 4.92 |
| CHEMBL1308389 | — | — | 1 | 4.90 |
| CHEMBL1588202 | — | — | 1 | 4.89 |
| CHEMBL1490069 | — | — | 1 | 4.84 |
| CHEMBL1719184 | — | — | 1 | 4.81 |
| CHEMBL1393837 | — | — | 1 | 4.81 |
| CHEMBL1440652 | — | — | 1 | 4.80 |
| CHEMBL1713166 | — | — | 1 | 4.77 |
| CHEMBL1429212 | — | — | 1 | 4.76 |
| CHEMBL1385823 | — | — | 1 | 4.76 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1732484 | — | EC50 | = | 502.9 | nM | 6.30 |
| CHEMBL1200531 | ALFENTANIL HYDROCHLORIDE | EC50 | = | 781.41 | nM | 6.11 |
| CHEMBL1717557 | — | EC50 | = | 1420.0 | nM | 5.85 |
| CHEMBL1463894 | — | EC50 | = | 2417.0 | nM | 5.62 |
| CHEMBL1307063 | — | EC50 | = | 2749.0 | nM | 5.56 |
| CHEMBL1331866 | — | EC50 | = | 2829.0 | nM | 5.55 |
| CHEMBL1581674 | — | EC50 | = | 3284.0 | nM | 5.48 |
| CHEMBL1700847 | — | EC50 | = | 3637.0 | nM | 5.44 |
| CHEMBL1380599 | — | EC50 | = | 4154.0 | nM | 5.38 |
| CHEMBL1388222 | — | EC50 | = | 4670.0 | nM | 5.33 |
| CHEMBL1416425 | — | EC50 | = | 4641.0 | nM | 5.33 |
| CHEMBL1522542 | — | EC50 | = | 4846.0 | nM | 5.32 |
| CHEMBL1609119 | — | EC50 | = | 5100.0 | nM | 5.29 |
| CHEMBL542581 | PHENCYCLIDINE HYDROCHLORIDE | EC50 | = | 6290.0 | nM | 5.20 |
| CHEMBL1698841 | — | EC50 | = | 7495.0 | nM | 5.12 |
| CHEMBL1531675 | — | EC50 | = | 10097.0 | nM | 5.00 |
| CHEMBL1426979 | — | EC50 | = | 10277.0 | nM | 4.99 |
| CHEMBL1460676 | — | EC50 | = | 10199.0 | nM | 4.99 |
| CHEMBL1586285 | — | EC50 | = | 10799.0 | nM | 4.97 |
| CHEMBL1705302 | — | EC50 | = | 10948.0 | nM | 4.96 |
| CHEMBL1720091 | — | EC50 | = | 12037.0 | nM | 4.92 |
| CHEMBL1308389 | — | EC50 | = | 12489.0 | nM | 4.90 |
| CHEMBL1588202 | — | EC50 | = | 12955.0 | nM | 4.89 |
| CHEMBL1490069 | — | EC50 | = | 14489.0 | nM | 4.84 |
| CHEMBL1719184 | — | EC50 | = | 15641.0 | nM | 4.81 |
| CHEMBL1393837 | — | EC50 | = | 15497.0 | nM | 4.81 |
| CHEMBL1440652 | — | EC50 | = | 15708.0 | nM | 4.80 |
| CHEMBL1713166 | — | EC50 | = | 17060.0 | nM | 4.77 |
| CHEMBL1385823 | — | EC50 | = | 17520.0 | nM | 4.76 |
| CHEMBL1429212 | — | EC50 | = | 17286.0 | nM | 4.76 |
| CHEMBL1315401 | — | EC50 | = | 17999.0 | nM | 4.75 |
| CHEMBL1425453 | — | EC50 | = | 18742.0 | nM | 4.73 |
| CHEMBL1709988 | — | EC50 | = | 18532.0 | nM | 4.73 |
| CHEMBL1448229 | — | EC50 | = | 18886.0 | nM | 4.72 |
| CHEMBL1902708 | — | EC50 | = | 20825.0 | nM | 4.68 |
| CHEMBL1473706 | — | EC50 | = | 22850.0 | nM | 4.64 |
| CHEMBL1612697 | — | EC50 | = | 24291.0 | nM | 4.62 |
| CHEMBL1581275 | — | EC50 | = | 24758.0 | nM | 4.61 |
| CHEMBL1356740 | — | EC50 | = | 26278.0 | nM | 4.58 |
| CHEMBL1407554 | — | EC50 | = | 26183.0 | nM | 4.58 |
| CHEMBL1412340 | — | EC50 | = | 29206.0 | nM | 4.54 |
| CHEMBL1566963 | — | EC50 | = | 33448.0 | nM | 4.48 |
| CHEMBL1422217 | — | EC50 | = | 35107.0 | nM | 4.46 |
| CHEMBL1584594 | — | EC50 | = | 36748.0 | nM | 4.43 |
| CHEMBL1513567 | — | EC50 | = | 40636.0 | nM | 4.39 |
| CHEMBL1533638 | — | EC50 | = | 42974.0 | nM | 4.37 |
| CHEMBL1587574 | — | EC50 | = | 42765.0 | nM | 4.37 |
| CHEMBL3213958 | — | EC50 | = | 42819.0 | nM | 4.37 |
| CHEMBL1423609 | — | EC50 | = | 43874.0 | nM | 4.36 |
| CHEMBL1198307 | — | EC50 | = | 43795.0 | nM | 4.36 |