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Assay Detail

CHEMBL1909170

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
DRUGMATRIX: Muscarinic M1 radioligand binding (ligand: [3H] N-Methylscopolamine)
1742
Total Activities
871
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Cell Type CHO-K1
Subcellular Membrane
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Muscarinic acetylcholine receptor M1 (CHEMBL216)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

DrugMatrix in vitro pharmacology data
Scott S. Auerbach, DrugMatrix¨ and ToxFX¨ Coordinator National Toxicology Program

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 871 6.38 9.26
Ki 871 7.00 9.88

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1201203 BENZTROPINE 4.0 2 9.88
CHEMBL1354199 METHSCOPOLAMINE BROMIDE 4.0 2 9.49
CHEMBL517712 ATROPINE 4.0 2 9.44
CHEMBL1123 DICYCLOMINE 4.0 2 9.08
CHEMBL1231 OXYBUTYNIN 4.0 2 9.07
CHEMBL1490 TRIHEXYPHENIDYL 4.0 2 8.87
CHEMBL479 THIORIDAZINE 4.0 2 8.77
CHEMBL42 CLOZAPINE 4.0 2 8.61
CHEMBL629 AMITRIPTYLINE 4.0 2 8.56
CHEMBL2107687 VALETHAMATE BROMIDE -1.0 2 8.56
CHEMBL643 PROMETHAZINE 4.0 2 8.48
CHEMBL516 CYPROHEPTADINE 4.0 2 8.40
CHEMBL334255 CETYLPYRIDINIUM BROMIDE 2 8.10
CHEMBL1909073 PIPERILATE ETHOBROMIDE 2 8.08
CHEMBL1628227 DOXEPIN 4.0 2 7.75
CHEMBL395110 MEPAZINE 4.0 2 7.72
CHEMBL71 CHLORPROMAZINE 4.0 2 7.70
CHEMBL445 NORTRIPTYLINE 4.0 2 7.70
CHEMBL415 CLOMIPRAMINE 4.0 2 7.66
CHEMBL1319362 HOMATROPINE HYDROBROMIDE -1.0 2 7.50
CHEMBL490 PAROXETINE 4.0 2 7.46
CHEMBL900 ORPHENADRINE 4.0 2 7.44
CHEMBL1172 DESLORATADINE 4.0 2 7.19
CHEMBL1200604 TROPICAMIDE 4.0 2 7.17
CHEMBL936 DIPHENIDOL 4.0 2 7.11
CHEMBL657 DIPHENHYDRAMINE 4.0 2 7.08
CHEMBL221753 BENZETHONIUM CHLORIDE 2.0 2 7.00
CHEMBL305660 EBASTINE 4.0 2 7.00
CHEMBL1200406 DIMENHYDRINATE 4.0 2 6.96
CHEMBL564 PROMAZINE 4.0 2 6.93

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1201203 BENZTROPINE Ki = 0.131 nM 9.88
CHEMBL1354199 METHSCOPOLAMINE BROMIDE Ki = 0.321 nM 9.49
CHEMBL517712 ATROPINE Ki = 0.366 nM 9.44
CHEMBL1201203 BENZTROPINE IC50 = 0.544 nM 9.26
CHEMBL1123 DICYCLOMINE Ki = 0.834 nM 9.08
CHEMBL1231 OXYBUTYNIN Ki = 0.847 nM 9.07
CHEMBL1354199 METHSCOPOLAMINE BROMIDE IC50 = 1.334 nM 8.88
CHEMBL1490 TRIHEXYPHENIDYL Ki = 1.351 nM 8.87
CHEMBL517712 ATROPINE IC50 = 1.521 nM 8.82
CHEMBL479 THIORIDAZINE Ki = 1.69 nM 8.77
CHEMBL42 CLOZAPINE Ki = 2.474 nM 8.61
CHEMBL629 AMITRIPTYLINE Ki = 2.724 nM 8.56
CHEMBL2107687 VALETHAMATE BROMIDE Ki = 2.78 nM 8.56
CHEMBL643 PROMETHAZINE Ki = 3.321 nM 8.48
CHEMBL1123 DICYCLOMINE IC50 = 3.463 nM 8.46
CHEMBL1231 OXYBUTYNIN IC50 = 3.518 nM 8.45
CHEMBL516 CYPROHEPTADINE Ki = 3.943 nM 8.40
CHEMBL1490 TRIHEXYPHENIDYL IC50 = 5.608 nM 8.25
CHEMBL479 THIORIDAZINE IC50 = 7.019 nM 8.15
CHEMBL334255 CETYLPYRIDINIUM BROMIDE Ki = 7.941 nM 8.10
CHEMBL1909073 PIPERILATE ETHOBROMIDE Ki = 8.387 nM 8.08
CHEMBL42 CLOZAPINE IC50 = 10.0 nM 8.00
CHEMBL629 AMITRIPTYLINE IC50 = 11.0 nM 7.96
CHEMBL2107687 VALETHAMATE BROMIDE IC50 = 12.0 nM 7.92
CHEMBL643 PROMETHAZINE IC50 = 14.0 nM 7.85
CHEMBL516 CYPROHEPTADINE IC50 = 16.0 nM 7.80
CHEMBL1628227 DOXEPIN Ki = 18.0 nM 7.75
CHEMBL395110 MEPAZINE Ki = 19.0 nM 7.72
CHEMBL71 CHLORPROMAZINE Ki = 20.0 nM 7.70
CHEMBL445 NORTRIPTYLINE Ki = 20.0 nM 7.70
CHEMBL415 CLOMIPRAMINE Ki = 22.0 nM 7.66
CHEMBL1319362 HOMATROPINE HYDROBROMIDE Ki = 32.0 nM 7.50
CHEMBL334255 CETYLPYRIDINIUM BROMIDE IC50 = 33.0 nM 7.48
CHEMBL490 PAROXETINE Ki = 35.0 nM 7.46
CHEMBL1909073 PIPERILATE ETHOBROMIDE IC50 = 35.0 nM 7.46
CHEMBL900 ORPHENADRINE Ki = 36.0 nM 7.44
CHEMBL1172 DESLORATADINE Ki = 64.0 nM 7.19
CHEMBL1200604 TROPICAMIDE Ki = 68.0 nM 7.17
CHEMBL936 DIPHENIDOL Ki = 78.0 nM 7.11
CHEMBL1628227 DOXEPIN IC50 = 77.0 nM 7.11
CHEMBL395110 MEPAZINE IC50 = 79.0 nM 7.10
CHEMBL445 NORTRIPTYLINE IC50 = 82.0 nM 7.09
CHEMBL71 CHLORPROMAZINE IC50 = 83.0 nM 7.08
CHEMBL657 DIPHENHYDRAMINE Ki = 83.0 nM 7.08
CHEMBL415 CLOMIPRAMINE IC50 = 91.0 nM 7.04
CHEMBL305660 EBASTINE Ki = 101.2 nM 7.00
CHEMBL221753 BENZETHONIUM CHLORIDE Ki = 99.0 nM 7.00
CHEMBL1200406 DIMENHYDRINATE Ki = 109.0 nM 6.96
CHEMBL564 PROMAZINE Ki = 117.0 nM 6.93
CHEMBL1319362 HOMATROPINE HYDROBROMIDE IC50 = 131.0 nM 6.88