Assay Detail
Functional
CHEMBL1963969
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for inhibitors of the Steroid Receptor Coactivator 1 (SRC1; NCOA1): Luminescence-based cell-based high throughput dose response assay to identify inhibitors of the Steroid Receptor Coactivator 3 (SRC3; NCOA3). (Class of assay: confirmatory)
240
Total Activities
240
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 240 | 5.32 | 7.73 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL132431 | — | — | 1 | 7.73 |
| CHEMBL1571037 | — | — | 1 | 7.04 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 6.68 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.43 |
| CHEMBL1699187 | — | — | 1 | 6.36 |
| CHEMBL1373969 | — | — | 1 | 6.30 |
| CHEMBL1705854 | — | — | 1 | 6.28 |
| CHEMBL1713127 | — | — | 1 | 6.18 |
| CHEMBL1611106 | — | — | 1 | 6.16 |
| CHEMBL1306377 | — | — | 1 | 6.12 |
| CHEMBL59530 | — | — | 1 | 6.02 |
| CHEMBL1713613 | — | — | 1 | 6.00 |
| CHEMBL1444434 | — | — | 1 | 5.99 |
| CHEMBL1445386 | — | — | 1 | 5.98 |
| CHEMBL1475299 | — | — | 1 | 5.97 |
| CHEMBL1302818 | — | — | 1 | 5.97 |
| CHEMBL1413178 | — | — | 1 | 5.92 |
| CHEMBL1608402 | — | — | 1 | 5.89 |
| CHEMBL1200512 | IRINOTECAN HYDROCHLORIDE HYDRATE | — | 1 | 5.88 |
| CHEMBL1612809 | — | — | 1 | 5.86 |
| CHEMBL1307972 | — | — | 1 | 5.86 |
| CHEMBL1383315 | — | — | 1 | 5.84 |
| CHEMBL1370927 | — | — | 1 | 5.80 |
| CHEMBL1469670 | — | — | 1 | 5.80 |
| CHEMBL1418980 | — | — | 1 | 5.76 |
| CHEMBL1399772 | — | — | 1 | 5.68 |
| CHEMBL1965654 | — | — | 1 | 5.68 |
| CHEMBL1421781 | — | — | 1 | 5.67 |
| CHEMBL1412433 | — | — | 1 | 5.67 |
| CHEMBL1400379 | — | — | 1 | 5.67 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL132431 | — | IC50 | = | 18.61 | nM | 7.73 |
| CHEMBL1571037 | — | IC50 | = | 91.26 | nM | 7.04 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 210.97 | nM | 6.68 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 374.72 | nM | 6.43 |
| CHEMBL1699187 | — | IC50 | = | 434.07 | nM | 6.36 |
| CHEMBL1373969 | — | IC50 | = | 503.09 | nM | 6.30 |
| CHEMBL1705854 | — | IC50 | = | 521.85 | nM | 6.28 |
| CHEMBL1713127 | — | IC50 | = | 660.61 | nM | 6.18 |
| CHEMBL1611106 | — | IC50 | = | 694.34 | nM | 6.16 |
| CHEMBL1306377 | — | IC50 | = | 762.3 | nM | 6.12 |
| CHEMBL59530 | — | IC50 | = | 950.0 | nM | 6.02 |
| CHEMBL1713613 | — | IC50 | = | 1008.0 | nM | 6.00 |
| CHEMBL1444434 | — | IC50 | = | 1016.0 | nM | 5.99 |
| CHEMBL1445386 | — | IC50 | = | 1049.0 | nM | 5.98 |
| CHEMBL1475299 | — | IC50 | = | 1077.0 | nM | 5.97 |
| CHEMBL1302818 | — | IC50 | = | 1072.0 | nM | 5.97 |
| CHEMBL1413178 | — | IC50 | = | 1197.0 | nM | 5.92 |
| CHEMBL1608402 | — | IC50 | = | 1279.0 | nM | 5.89 |
| CHEMBL1200512 | IRINOTECAN HYDROCHLORIDE HYDRATE | IC50 | = | 1315.0 | nM | 5.88 |
| CHEMBL1612809 | — | IC50 | = | 1378.0 | nM | 5.86 |
| CHEMBL1307972 | — | IC50 | = | 1386.0 | nM | 5.86 |
| CHEMBL1383315 | — | IC50 | = | 1444.0 | nM | 5.84 |
| CHEMBL1469670 | — | IC50 | = | 1583.0 | nM | 5.80 |
| CHEMBL1370927 | — | IC50 | = | 1575.0 | nM | 5.80 |
| CHEMBL1418980 | — | IC50 | = | 1744.0 | nM | 5.76 |
| CHEMBL1399772 | — | IC50 | = | 2090.0 | nM | 5.68 |
| CHEMBL1965654 | — | IC50 | = | 2091.0 | nM | 5.68 |
| CHEMBL1412433 | — | IC50 | = | 2136.0 | nM | 5.67 |
| CHEMBL1400379 | — | IC50 | = | 2116.0 | nM | 5.67 |
| CHEMBL1421781 | — | IC50 | = | 2128.0 | nM | 5.67 |
| CHEMBL494325 | — | IC50 | = | 2299.0 | nM | 5.64 |
| CHEMBL1502254 | — | IC50 | = | 2458.0 | nM | 5.61 |
| CHEMBL2005690 | — | IC50 | = | 2568.0 | nM | 5.59 |
| CHEMBL1456725 | — | IC50 | = | 2621.0 | nM | 5.58 |
| CHEMBL1535999 | — | IC50 | = | 2634.0 | nM | 5.58 |
| CHEMBL1528507 | — | IC50 | = | 2615.0 | nM | 5.58 |
| CHEMBL1471916 | — | IC50 | = | 2695.0 | nM | 5.57 |
| CHEMBL1398705 | — | IC50 | = | 2669.0 | nM | 5.57 |
| CHEMBL1610875 | — | IC50 | = | 2751.0 | nM | 5.56 |
| CHEMBL1318140 | — | IC50 | = | 2810.0 | nM | 5.55 |
| CHEMBL533226 | — | IC50 | = | 2893.0 | nM | 5.54 |
| CHEMBL1469961 | — | IC50 | = | 2870.0 | nM | 5.54 |
| CHEMBL356169 | — | IC50 | = | 2991.0 | nM | 5.52 |
| CHEMBL1406398 | — | IC50 | = | 3108.0 | nM | 5.51 |
| CHEMBL1368216 | — | IC50 | = | 3109.0 | nM | 5.51 |
| CHEMBL1480880 | — | IC50 | = | 3161.0 | nM | 5.50 |
| CHEMBL1605666 | — | IC50 | = | 3211.0 | nM | 5.49 |
| CHEMBL1899898 | — | IC50 | = | 3276.0 | nM | 5.49 |
| CHEMBL1453181 | — | IC50 | = | 3234.0 | nM | 5.49 |
| CHEMBL1427335 | — | IC50 | = | 3236.0 | nM | 5.49 |