Assay Detail
Functional
CHEMBL2363173
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SANGER: Inhibition of human D-566MG cell growth in a cell viability assay.
61
Total Activities
61
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | D-566MG |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 61 | 5.73 | 9.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.88 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.74 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.69 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 8.41 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 8.14 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.82 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.75 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 7.02 |
| CHEMBL217354 | — | — | 1 | 6.94 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.83 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.57 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.08 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.97 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.90 |
| CHEMBL577784 | BX-795 | — | 1 | 5.88 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 5.85 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 5.80 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 5.79 |
| CHEMBL202721 | — | — | 1 | 5.75 |
| CHEMBL521686 | OLAPARIB | 4.0 | 1 | 5.61 |
| CHEMBL573107 | — | — | 1 | 5.54 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 1 | 5.51 |
| CHEMBL379975 | — | — | 1 | 5.49 |
| CHEMBL11359 | CISPLATIN | 4.0 | 1 | 5.46 |
| CHEMBL3349342 | — | — | 1 | 5.37 |
| CHEMBL2137530 | SERDEMETAN | 2.0 | 1 | 5.20 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 5.18 |
| CHEMBL393929 | — | — | 1 | 5.17 |
| CHEMBL255863 | NILOTINIB | 4.0 | 1 | 5.13 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 5.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.1315 | nM | 9.88 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.1823 | nM | 9.74 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 2.043 | nM | 8.69 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 3.904 | nM | 8.41 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 7.157 | nM | 8.14 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 15.23 | nM | 7.82 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 17.69 | nM | 7.75 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 96.46 | nM | 7.02 |
| CHEMBL217354 | — | IC50 | = | 115.75 | nM | 6.94 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 146.9 | nM | 6.83 |
| CHEMBL803 | CYTARABINE | IC50 | = | 269.04 | nM | 6.57 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 838.62 | nM | 6.08 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1067.26 | nM | 5.97 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 1252.89 | nM | 5.90 |
| CHEMBL577784 | BX-795 | IC50 | = | 1304.48 | nM | 5.88 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 1406.83 | nM | 5.85 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1571.55 | nM | 5.80 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 1625.3 | nM | 5.79 |
| CHEMBL202721 | — | IC50 | = | 1787.75 | nM | 5.75 |
| CHEMBL521686 | OLAPARIB | IC50 | = | 2445.68 | nM | 5.61 |
| CHEMBL573107 | — | IC50 | = | 2912.95 | nM | 5.54 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 3073.74 | nM | 5.51 |
| CHEMBL379975 | — | IC50 | = | 3271.58 | nM | 5.49 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 3476.48 | nM | 5.46 |
| CHEMBL3349342 | — | IC50 | = | 4265.77 | nM | 5.37 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 6334.91 | nM | 5.20 |
| CHEMBL105442 | CI-1040 | IC50 | = | 6543.03 | nM | 5.18 |
| CHEMBL393929 | — | IC50 | = | 6788.73 | nM | 5.17 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 7471.55 | nM | 5.13 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 8044.29 | nM | 5.09 |
| CHEMBL939 | GEFITINIB | IC50 | = | 9018.1 | nM | 5.04 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 9836.64 | nM | 5.01 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 13957.58 | nM | 4.86 |
| CHEMBL102714 | SB-216763 | IC50 | = | 13948.07 | nM | 4.86 |
| CHEMBL188678 | — | IC50 | = | 14770.62 | nM | 4.83 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 16726.24 | nM | 4.78 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 20588.84 | nM | 4.69 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 21868.98 | nM | 4.66 |
| CHEMBL189584 | PD-173074 | IC50 | = | 22760.08 | nM | 4.64 |
| CHEMBL473417 | VISMODEGIB | IC50 | = | 25294.32 | nM | 4.60 |
| CHEMBL477989 | SB590885 | IC50 | = | 27192.85 | nM | 4.57 |
| CHEMBL399530 | — | IC50 | = | 26887.86 | nM | 4.57 |
| CHEMBL1090090 | VX-702 | IC50 | = | 29217.59 | nM | 4.53 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 29939.3 | nM | 4.52 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 41208.6 | nM | 4.38 |
| CHEMBL222102 | KU-55933 | IC50 | = | 49909.63 | nM | 4.30 |
| CHEMBL2134202 | — | IC50 | = | 63522.36 | nM | 4.20 |
| CHEMBL38 | TRETINOIN | IC50 | = | 89594.42 | nM | 4.05 |
| CHEMBL506871 | VELIPARIB | IC50 | = | 96230.75 | nM | 4.02 |
| CHEMBL848 | LENALIDOMIDE | IC50 | = | 107635.12 | nM | - |