Assay Detail
Functional
CHEMBL2363215
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SANGER: Inhibition of human ES7 cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | ES7 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.70 | 10.59 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 10.59 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.41 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.12 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.45 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 8.44 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.41 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.24 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.23 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.07 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.74 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.70 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.67 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.47 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.29 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.07 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 7.02 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 6.83 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.80 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.59 |
| CHEMBL217354 | — | — | 1 | 6.57 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.56 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.56 |
| CHEMBL585951 | — | — | 1 | 6.49 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.47 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.42 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.26 |
| CHEMBL300389 | — | — | 1 | 6.14 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.12 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 6.09 |
| CHEMBL577784 | BX-795 | — | 1 | 6.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.02543 | nM | 10.59 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.3885 | nM | 9.41 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.7663 | nM | 9.12 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 3.592 | nM | 8.45 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 3.653 | nM | 8.44 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 3.856 | nM | 8.41 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 5.753 | nM | 8.24 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 5.871 | nM | 8.23 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 8.457 | nM | 8.07 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 18.09 | nM | 7.74 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 19.76 | nM | 7.70 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 21.12 | nM | 7.67 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 33.74 | nM | 7.47 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 51.4 | nM | 7.29 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 85.85 | nM | 7.07 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 94.81 | nM | 7.02 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 148.36 | nM | 6.83 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 160.11 | nM | 6.80 |
| CHEMBL803 | CYTARABINE | IC50 | = | 257.16 | nM | 6.59 |
| CHEMBL217354 | — | IC50 | = | 270.34 | nM | 6.57 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 273.83 | nM | 6.56 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 273.09 | nM | 6.56 |
| CHEMBL585951 | — | IC50 | = | 324.55 | nM | 6.49 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 341.99 | nM | 6.47 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 377.54 | nM | 6.42 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 548.49 | nM | 6.26 |
| CHEMBL300389 | — | IC50 | = | 731.41 | nM | 6.14 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 767.13 | nM | 6.12 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 812.86 | nM | 6.09 |
| CHEMBL577784 | BX-795 | IC50 | = | 835.66 | nM | 6.08 |
| CHEMBL64925 | MG-132 | IC50 | = | 896.5 | nM | 6.05 |
| CHEMBL573107 | — | IC50 | = | 916.07 | nM | 6.04 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 936.38 | nM | 6.03 |
| CHEMBL1190711 | — | IC50 | = | 1087.55 | nM | 5.96 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 1113.34 | nM | 5.95 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 1295.42 | nM | 5.89 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 1279.51 | nM | 5.89 |
| CHEMBL258844 | — | IC50 | = | 1345.11 | nM | 5.87 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1474.09 | nM | 5.83 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 1538.48 | nM | 5.81 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1547.73 | nM | 5.81 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1803.02 | nM | 5.74 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 1874.13 | nM | 5.73 |
| CHEMBL191384 | — | IC50 | = | 3032.74 | nM | 5.52 |
| CHEMBL379975 | — | IC50 | = | 3015.14 | nM | 5.52 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 3255.84 | nM | 5.49 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 3399.11 | nM | 5.47 |
| CHEMBL188678 | — | IC50 | = | 3467.29 | nM | 5.46 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 5231.24 | nM | 5.28 |
| CHEMBL521686 | OLAPARIB | IC50 | = | 6035.77 | nM | 5.22 |