Assay Detail
Functional
CHEMBL2363676
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SANGER: Inhibition of human SW1088 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SW1088 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.51 | 8.53 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.53 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.24 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.77 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.56 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.55 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.50 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.35 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.10 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.08 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.79 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.49 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.47 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.35 |
| CHEMBL217354 | — | — | 1 | 6.34 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.27 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.16 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.06 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.04 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.99 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.93 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 5.89 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.87 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 5.78 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 5.71 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 5.70 |
| CHEMBL577784 | BX-795 | — | 1 | 5.70 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 5.68 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 5.60 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 5.56 |
| CHEMBL2137530 | SERDEMETAN | 2.0 | 1 | 5.55 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 2.948 | nM | 8.53 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 5.791 | nM | 8.24 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 16.97 | nM | 7.77 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 27.77 | nM | 7.56 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 28.29 | nM | 7.55 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 31.84 | nM | 7.50 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 44.9 | nM | 7.35 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 79.44 | nM | 7.10 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 82.14 | nM | 7.08 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 164.13 | nM | 6.79 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 324.04 | nM | 6.49 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 337.97 | nM | 6.47 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 443.9 | nM | 6.35 |
| CHEMBL217354 | — | IC50 | = | 454.6 | nM | 6.34 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 538.69 | nM | 6.27 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 699.55 | nM | 6.16 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 873.73 | nM | 6.06 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 915.52 | nM | 6.04 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 1030.55 | nM | 5.99 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1168.79 | nM | 5.93 |
| CHEMBL939 | GEFITINIB | IC50 | = | 1296.07 | nM | 5.89 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1366.12 | nM | 5.87 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 1661.67 | nM | 5.78 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 1946.06 | nM | 5.71 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 2014.76 | nM | 5.70 |
| CHEMBL577784 | BX-795 | IC50 | = | 1996.73 | nM | 5.70 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 2069.31 | nM | 5.68 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 2481.43 | nM | 5.61 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 2492.13 | nM | 5.60 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 2778.39 | nM | 5.56 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 2806.51 | nM | 5.55 |
| CHEMBL803 | CYTARABINE | IC50 | = | 3313.61 | nM | 5.48 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 3474.7 | nM | 5.46 |
| CHEMBL572881 | MOTESANIB | IC50 | = | 4395.25 | nM | 5.36 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 4668.27 | nM | 5.33 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 5029.44 | nM | 5.30 |
| CHEMBL135561 | — | IC50 | = | 5160.76 | nM | 5.29 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 6443.97 | nM | 5.19 |
| CHEMBL105442 | CI-1040 | IC50 | = | 6919.13 | nM | 5.16 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 7658.26 | nM | 5.12 |
| CHEMBL3349342 | — | IC50 | = | 7518.56 | nM | 5.12 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 8569.21 | nM | 5.07 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 9560.98 | nM | 5.02 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 9699.31 | nM | 5.01 |
| CHEMBL202721 | — | IC50 | = | 10354.01 | nM | 4.99 |
| CHEMBL2363137 | — | IC50 | = | 12254.58 | nM | 4.91 |
| CHEMBL379975 | — | IC50 | = | 15554.31 | nM | 4.81 |
| CHEMBL221137 | EMBELIN | IC50 | = | 16654.73 | nM | 4.78 |
| CHEMBL512504 | — | IC50 | = | 19944.73 | nM | 4.70 |
| CHEMBL210618 | — | IC50 | = | 23164.08 | nM | 4.63 |