Assay Detail
Functional
CHEMBL2363772
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SANGER: Inhibition of human C32 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | C32 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.61 | 8.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 8.52 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 8.44 |
| CHEMBL2363137 | — | — | 1 | 8.17 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.87 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.58 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.33 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.27 |
| CHEMBL3349342 | — | — | 1 | 7.24 |
| CHEMBL1614701 | SELUMETINIB | 4.0 | 1 | 7.01 |
| CHEMBL477989 | SB590885 | — | 1 | 7.00 |
| CHEMBL1230020 | PLX-4720 | — | 1 | 6.82 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.74 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 6.72 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.51 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.46 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.38 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.34 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.24 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.14 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 6.13 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 6.06 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 5.95 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 5.92 |
| CHEMBL379975 | — | — | 1 | 5.82 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 5.82 |
| CHEMBL577784 | BX-795 | — | 1 | 5.75 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 5.72 |
| CHEMBL217354 | — | — | 1 | 5.70 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.57 |
| CHEMBL221137 | EMBELIN | — | 1 | 5.55 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 3.045 | nM | 8.52 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 3.668 | nM | 8.44 |
| CHEMBL2363137 | — | IC50 | = | 6.742 | nM | 8.17 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 13.37 | nM | 7.87 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 26.3 | nM | 7.58 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 46.64 | nM | 7.33 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 53.83 | nM | 7.27 |
| CHEMBL3349342 | — | IC50 | = | 57.17 | nM | 7.24 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 98.23 | nM | 7.01 |
| CHEMBL477989 | SB590885 | IC50 | = | 99.63 | nM | 7.00 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 151.31 | nM | 6.82 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 181.88 | nM | 6.74 |
| CHEMBL105442 | CI-1040 | IC50 | = | 190.72 | nM | 6.72 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 309.46 | nM | 6.51 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 346.82 | nM | 6.46 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 419.28 | nM | 6.38 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 452.29 | nM | 6.34 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 573.13 | nM | 6.24 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 724.84 | nM | 6.14 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 741.12 | nM | 6.13 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 866.85 | nM | 6.06 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 1118.24 | nM | 5.95 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 1190.88 | nM | 5.92 |
| CHEMBL379975 | — | IC50 | = | 1530.32 | nM | 5.82 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 1528.34 | nM | 5.82 |
| CHEMBL577784 | BX-795 | IC50 | = | 1763.9 | nM | 5.75 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 1912.59 | nM | 5.72 |
| CHEMBL217354 | — | IC50 | = | 2015.95 | nM | 5.70 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 2677.89 | nM | 5.57 |
| CHEMBL221137 | EMBELIN | IC50 | = | 2825.82 | nM | 5.55 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 2924.7 | nM | 5.53 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 3415.08 | nM | 5.47 |
| CHEMBL202721 | — | IC50 | = | 3828.98 | nM | 5.42 |
| CHEMBL573107 | — | IC50 | = | 3965.81 | nM | 5.40 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 5600.29 | nM | 5.25 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 6130.34 | nM | 5.21 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 6376.66 | nM | 5.20 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 8533.84 | nM | 5.07 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 8439.27 | nM | 5.07 |
| CHEMBL572881 | MOTESANIB | IC50 | = | 8784.42 | nM | 5.06 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 9330.64 | nM | 5.03 |
| CHEMBL939 | GEFITINIB | IC50 | = | 9633.4 | nM | 5.02 |
| CHEMBL188678 | — | IC50 | = | 10834.74 | nM | 4.96 |
| CHEMBL803 | CYTARABINE | IC50 | = | 13274.53 | nM | 4.88 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 16971.68 | nM | 4.77 |
| CHEMBL240954 | — | IC50 | = | 17660.56 | nM | 4.75 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 18472.74 | nM | 4.73 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 19045.05 | nM | 4.72 |
| CHEMBL585951 | — | IC50 | = | 21120.96 | nM | 4.67 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 21863.51 | nM | 4.66 |