Assay Detail
Functional
CHEMBL2363826
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human YH-13 cell growth in a cell viability assay.
61
Total Activities
61
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | YH-13 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 61 | 5.67 | 9.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.10 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.43 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.93 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.66 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.62 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.39 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.24 |
| CHEMBL217354 | — | — | 1 | 7.15 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.87 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.80 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.52 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.49 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.26 |
| CHEMBL577784 | BX-795 | — | 1 | 6.20 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.90 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.82 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 1 | 5.71 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 5.65 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 5.61 |
| CHEMBL3349342 | — | — | 1 | 5.57 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 5.46 |
| CHEMBL188678 | — | — | 1 | 5.41 |
| CHEMBL393929 | — | — | 1 | 5.32 |
| CHEMBL572881 | MOTESANIB | 3.0 | 1 | 5.10 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 5.07 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 4.99 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 4.95 |
| CHEMBL573107 | — | — | 1 | 4.94 |
| CHEMBL11359 | CISPLATIN | 4.0 | 1 | 4.92 |
| CHEMBL189584 | PD-173074 | — | 1 | 4.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.7908 | nM | 9.10 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 3.702 | nM | 8.43 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 11.65 | nM | 7.93 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 21.88 | nM | 7.66 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 24.15 | nM | 7.62 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 41.08 | nM | 7.39 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 57.22 | nM | 7.24 |
| CHEMBL217354 | — | IC50 | = | 70.59 | nM | 7.15 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 134.54 | nM | 6.87 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 156.74 | nM | 6.80 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 304.32 | nM | 6.52 |
| CHEMBL803 | CYTARABINE | IC50 | = | 327.55 | nM | 6.49 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 549.38 | nM | 6.26 |
| CHEMBL577784 | BX-795 | IC50 | = | 628.88 | nM | 6.20 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 1246.08 | nM | 5.90 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1498.94 | nM | 5.82 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1945.48 | nM | 5.71 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 2216.71 | nM | 5.65 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 2461.53 | nM | 5.61 |
| CHEMBL3349342 | — | IC50 | = | 2680.0 | nM | 5.57 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 3440.79 | nM | 5.46 |
| CHEMBL188678 | — | IC50 | = | 3871.89 | nM | 5.41 |
| CHEMBL393929 | — | IC50 | = | 4757.76 | nM | 5.32 |
| CHEMBL572881 | MOTESANIB | IC50 | = | 8006.22 | nM | 5.10 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 8610.08 | nM | 5.07 |
| CHEMBL939 | GEFITINIB | IC50 | = | 10305.66 | nM | 4.99 |
| CHEMBL105442 | CI-1040 | IC50 | = | 11326.73 | nM | 4.95 |
| CHEMBL573107 | — | IC50 | = | 11474.19 | nM | 4.94 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 12132.77 | nM | 4.92 |
| CHEMBL189584 | PD-173074 | IC50 | = | 12034.63 | nM | 4.92 |
| CHEMBL102714 | SB-216763 | IC50 | = | 16686.5 | nM | 4.78 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 20891.95 | nM | 4.68 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 21406.55 | nM | 4.67 |
| CHEMBL222102 | KU-55933 | IC50 | = | 22512.3 | nM | 4.65 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 33253.5 | nM | 4.48 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 35919.99 | nM | 4.45 |
| CHEMBL202721 | — | IC50 | = | 49422.12 | nM | 4.31 |
| CHEMBL1186585 | — | IC50 | = | 56348.47 | nM | 4.25 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 60046.84 | nM | 4.22 |
| CHEMBL521686 | OLAPARIB | IC50 | = | 64703.8 | nM | 4.19 |
| CHEMBL210618 | — | IC50 | = | 75845.77 | nM | 4.12 |
| CHEMBL176544 | — | IC50 | = | 89614.76 | nM | 4.05 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 92891.86 | nM | 4.03 |
| CHEMBL477989 | SB590885 | IC50 | = | 722578.45 | nM | - |
| CHEMBL255342 | — | IC50 | = | 591207.47 | nM | - |
| CHEMBL399530 | — | IC50 | = | 393568.45 | nM | - |
| CHEMBL1090771 | AVAGACESTAT | IC50 | = | 508580.75 | nM | - |
| CHEMBL2134202 | — | IC50 | = | 173134.37 | nM | - |
| CHEMBL1431 | METFORMIN | IC50 | = | 28266114.54 | nM | - |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 126006.69 | nM | - |