Assay Detail
Functional
CHEMBL3215070
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PubChem BioAssay. SAR analysis of small molecule antagonists of Gli-SUFU in a luminescent reporter assay - Set 2. (Class of assay: confirmatory)
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 28 | 7.15 | 7.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1393367 | — | — | 1 | 7.64 |
| CHEMBL3187872 | — | — | 1 | 7.62 |
| CHEMBL1438842 | — | — | 1 | 7.57 |
| CHEMBL3184876 | — | — | 1 | 7.46 |
| CHEMBL1523428 | — | — | 1 | 5.47 |
| CHEMBL3182177 | — | — | 1 | - |
| CHEMBL3182201 | — | — | 1 | - |
| CHEMBL3182548 | — | — | 1 | - |
| CHEMBL3182703 | — | — | 1 | - |
| CHEMBL3183417 | — | — | 1 | - |
| CHEMBL3183804 | — | — | 1 | - |
| CHEMBL3183962 | — | — | 1 | - |
| CHEMBL3184558 | — | — | 1 | - |
| CHEMBL3184611 | — | — | 1 | - |
| CHEMBL1583316 | — | — | 1 | - |
| CHEMBL3185202 | — | — | 1 | - |
| CHEMBL3182163 | — | — | 1 | - |
| CHEMBL3185857 | — | — | 1 | - |
| CHEMBL3186476 | — | — | 1 | - |
| CHEMBL3186610 | — | — | 1 | - |
| CHEMBL3187121 | — | — | 1 | - |
| CHEMBL3187241 | — | — | 1 | - |
| CHEMBL3187493 | — | — | 1 | - |
| CHEMBL3187538 | — | — | 1 | - |
| CHEMBL3187814 | — | — | 1 | - |
| CHEMBL3187975 | — | — | 1 | - |
| CHEMBL3188297 | — | — | 1 | - |
| CHEMBL3185694 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1393367 | — | IC50 | = | 23.0 | nM | 7.64 |
| CHEMBL3187872 | — | IC50 | = | 24.0 | nM | 7.62 |
| CHEMBL1438842 | — | IC50 | = | 27.0 | nM | 7.57 |
| CHEMBL3184876 | — | IC50 | = | 35.0 | nM | 7.46 |
| CHEMBL1523428 | — | IC50 | = | 3402.0 | nM | 5.47 |
| CHEMBL3182177 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3182201 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3182548 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3182703 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3183417 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3183804 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3183962 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3184558 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3184611 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL1583316 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3185202 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3182163 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3185857 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3186476 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3186610 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3187121 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3187241 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3187493 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3187538 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3187814 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3187975 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3188297 | — | IC50 | > | 9700.0 | nM | - |
| CHEMBL3185694 | — | IC50 | > | 9700.0 | nM | - |