Assay Detail
Binding
CHEMBL3419224
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Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assay
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Bromodomain adjacent to zinc finger domain protein 2A (CHEMBL3108642) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Structure enabled design of BAZ2-ICR, a chemical probe targeting the bromodomains of BAZ2A and BAZ2B.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 12 | 5.77 | 6.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4296718 | — | — | 1 | 6.89 |
| CHEMBL3415185 | — | — | 1 | 6.35 |
| CHEMBL3415182 | — | — | 1 | 6.22 |
| CHEMBL3415184 | — | — | 1 | 6.00 |
| CHEMBL3415186 | — | — | 1 | 5.86 |
| CHEMBL3415177 | — | — | 1 | 5.40 |
| CHEMBL3415179 | — | — | 1 | 5.11 |
| CHEMBL3415176 | — | — | 1 | 4.29 |
| CHEMBL3415183 | — | — | 1 | - |
| CHEMBL3415181 | — | — | 1 | - |
| CHEMBL3415180 | — | — | 1 | - |
| CHEMBL3415178 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4296718 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL3415185 | — | IC50 | = | 450.0 | nM | 6.35 |
| CHEMBL3415182 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3415184 | — | IC50 | = | 1010.0 | nM | 6.00 |
| CHEMBL3415186 | — | IC50 | = | 1380.0 | nM | 5.86 |
| CHEMBL3415177 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL3415179 | — | IC50 | = | 7800.0 | nM | 5.11 |
| CHEMBL3415176 | — | IC50 | = | 51000.0 | nM | 4.29 |
| CHEMBL3415183 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3415181 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3415180 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3415178 | — | IC50 | > | 50000.0 | nM | - |