Assay Detail
Functional
CHEMBL3562069
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PubChem BioAssay. Colo320 viability from Cell TiterGlo-IC50. (Class of assay: confirmatory)
234
Total Activities
233
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 234 | 6.14 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 9.00 |
| CHEMBL3182961 | — | — | 1 | 9.00 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | 4.0 | 2 | 9.00 |
| CHEMBL1394319 | BROQUINALDOL | 2.0 | 1 | 9.00 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | 4.0 | 1 | 9.00 |
| CHEMBL24944 | TRIBROMSALAN | 4.0 | 1 | 8.52 |
| CHEMBL1981438 | CLOFLUCARBAN | 2.0 | 1 | 8.52 |
| CHEMBL2360738 | — | — | 1 | 8.52 |
| CHEMBL232201 | BENZIODARONE | 4.0 | 1 | 8.52 |
| CHEMBL554041 | ALEXIDINE DIHYDROCHLORIDE | — | 1 | 8.39 |
| CHEMBL1448 | NICLOSAMIDE | 4.0 | 1 | 8.08 |
| CHEMBL290106 | BITHIONOL | 4.0 | 1 | 7.82 |
| CHEMBL1315136 | TIBROFAN | 2.0 | 1 | 7.75 |
| CHEMBL86754 | IODOQUINOL | 2.0 | 1 | 7.67 |
| CHEMBL50588 | EMETINE | 4.0 | 1 | 7.66 |
| CHEMBL1375045 | — | — | 1 | 7.43 |
| CHEMBL1200596 | CHLOROXINE | 4.0 | 1 | 7.31 |
| CHEMBL287542 | RAFOXANIDE | 2.0 | 1 | 7.27 |
| CHEMBL496 | HEXACHLOROPHENE | 4.0 | 1 | 7.24 |
| CHEMBL473535 | FENTICLOR | 2.0 | 1 | 7.12 |
| CHEMBL1320139 | HELIOMYCIN | 2.0 | 1 | 7.09 |
| CHEMBL12131 | CLOSANTEL | 2.0 | 1 | 6.94 |
| CHEMBL223448 | BROXYQUINOLINE | 4.0 | 1 | 6.94 |
| CHEMBL451887 | CARFILZOMIB | 4.0 | 1 | 6.84 |
| CHEMBL1788401 | CYCLOBENDAZOLE | 2.0 | 1 | 6.81 |
| CHEMBL1545634 | — | — | 1 | 6.79 |
| CHEMBL1450 | ATOVAQUONE | 4.0 | 1 | 6.75 |
| CHEMBL242580 | CICLOPIROX OLAMINE | 3.0 | 1 | 6.68 |
| CHEMBL1200398 | BUTOCONAZOLE NITRATE | 4.0 | 1 | 6.66 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL34259 | METHOTREXATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3182961 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1394319 | BROQUINALDOL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1981438 | CLOFLUCARBAN | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL232201 | BENZIODARONE | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL24944 | TRIBROMSALAN | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL2360738 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL554041 | ALEXIDINE DIHYDROCHLORIDE | IC50 | = | 4.1 | nM | 8.39 |
| CHEMBL1448 | NICLOSAMIDE | IC50 | = | 8.26 | nM | 8.08 |
| CHEMBL290106 | BITHIONOL | IC50 | = | 15.05 | nM | 7.82 |
| CHEMBL1315136 | TIBROFAN | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL86754 | IODOQUINOL | IC50 | = | 21.3 | nM | 7.67 |
| CHEMBL50588 | EMETINE | IC50 | = | 22.1 | nM | 7.66 |
| CHEMBL1375045 | — | IC50 | = | 37.2 | nM | 7.43 |
| CHEMBL1200596 | CHLOROXINE | IC50 | = | 49.33 | nM | 7.31 |
| CHEMBL287542 | RAFOXANIDE | IC50 | = | 54.0 | nM | 7.27 |
| CHEMBL496 | HEXACHLOROPHENE | IC50 | = | 57.2 | nM | 7.24 |
| CHEMBL473535 | FENTICLOR | IC50 | = | 74.99 | nM | 7.12 |
| CHEMBL1320139 | HELIOMYCIN | IC50 | = | 81.99 | nM | 7.09 |
| CHEMBL223448 | BROXYQUINOLINE | IC50 | = | 114.24 | nM | 6.94 |
| CHEMBL12131 | CLOSANTEL | IC50 | = | 116.0 | nM | 6.94 |
| CHEMBL451887 | CARFILZOMIB | IC50 | = | 144.59 | nM | 6.84 |
| CHEMBL1788401 | CYCLOBENDAZOLE | IC50 | = | 155.6 | nM | 6.81 |
| CHEMBL1545634 | — | IC50 | = | 160.8 | nM | 6.79 |
| CHEMBL1450 | ATOVAQUONE | IC50 | = | 176.4 | nM | 6.75 |
| CHEMBL242580 | CICLOPIROX OLAMINE | IC50 | = | 208.35 | nM | 6.68 |
| CHEMBL1200398 | BUTOCONAZOLE NITRATE | IC50 | = | 221.1 | nM | 6.66 |
| CHEMBL292009 | BUPARVAQUONE | IC50 | = | 254.8 | nM | 6.59 |
| CHEMBL3185933 | IODOPHTHALEIN SODIUM | IC50 | = | 311.53 | nM | 6.51 |
| CHEMBL388676 | CAPTAN | IC50 | = | 305.7 | nM | 6.51 |
| CHEMBL417799 | SANGUINARIUM | IC50 | = | 349.8 | nM | 6.46 |
| CHEMBL1076347 | TRICLOCARBAN | IC50 | = | 361.67 | nM | 6.44 |
| CHEMBL727 | THIOGUANINE | IC50 | = | 372.99 | nM | 6.43 |
| CHEMBL2358886 | — | IC50 | = | 385.9 | nM | 6.41 |
| CHEMBL550348 | DEFERASIROX | IC50 | = | 408.51 | nM | 6.39 |
| CHEMBL2355158 | — | IC50 | = | 458.3 | nM | 6.34 |
| CHEMBL2359490 | — | IC50 | = | 466.19 | nM | 6.33 |
| CHEMBL1483 | ALBENDAZOLE | IC50 | = | 502.0 | nM | 6.30 |
| CHEMBL1200485 | SORAFENIB TOSYLATE | IC50 | = | 507.5 | nM | 6.29 |
| CHEMBL1569226 | — | IC50 | = | 530.12 | nM | 6.28 |
| CHEMBL81782 | — | IC50 | = | 561.99 | nM | 6.25 |
| CHEMBL497 | CLIOQUINOL | IC50 | = | 586.2 | nM | 6.23 |
| CHEMBL1413199 | DIPHENADIONE | IC50 | = | 621.11 | nM | 6.21 |
| CHEMBL316040 | TEPOXALIN | IC50 | = | 661.5 | nM | 6.18 |
| CHEMBL1454910 | NITROXOLINE | IC50 | = | 683.66 | nM | 6.17 |
| CHEMBL3188653 | — | IC50 | = | 735.4 | nM | 6.13 |