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Assay Detail

CHEMBL4182259

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Binding
Binding affinity to His-tagged BRD2 bromodomain 2 (unknown origin) by SPR assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Bromodomain-containing protein 2 (CHEMBL1293289)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Exploiting a water network to achieve enthalpy-driven, bromodomain-selective BET inhibitors.
Shadrick WR, Slavish PJ, Chai SC, Waddell B, Connelly M, Low JA, Tallant C, Young BM, Bharatham N, Knapp S, Boyd VA, Morfouace M, Roussel MF, Chen T, Lee RE, Kiplin Guy R, Shelat AA, Potter PM.
Bioorg Med Chem (2018) 26 : 25 -36
PubMed 29170024 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 7 7.10 7.33

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4209110 1 7.33
CHEMBL4205876 1 7.21
CHEMBL4210405 1 7.14
CHEMBL4202664 1 7.13
CHEMBL4206677 1 7.11
CHEMBL1957266 1 6.94
CHEMBL4207106 1 6.83

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4209110 Kd = 47.0 nM 7.33
CHEMBL4205876 Kd = 61.0 nM 7.21
CHEMBL4210405 Kd = 72.0 nM 7.14
CHEMBL4202664 Kd = 74.0 nM 7.13
CHEMBL4206677 Kd = 77.0 nM 7.11
CHEMBL1957266 Kd = 116.0 nM 6.94
CHEMBL4207106 Kd = 148.0 nM 6.83