Assay Detail
Binding
CHEMBL4307635
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysis
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Mitogen-activated protein kinase kinase kinase 14 (CHEMBL5888) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Structure Based Design of Potent Selective Inhibitors of Protein Kinase D1 (PKD1).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 16 | 8.25 | 9.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4524153 | — | — | 1 | 9.80 |
| CHEMBL4113471 | — | — | 1 | 9.10 |
| CHEMBL4109262 | — | — | 1 | 9.05 |
| CHEMBL4073390 | — | — | 1 | 9.00 |
| CHEMBL4111969 | — | — | 1 | 8.77 |
| CHEMBL4115120 | — | — | 1 | 8.51 |
| CHEMBL3692392 | — | — | 1 | 8.00 |
| CHEMBL3692489 | — | — | 1 | 7.85 |
| CHEMBL3978002 | — | — | 1 | 6.24 |
| CHEMBL4546659 | — | — | 1 | 6.20 |
| CHEMBL3896516 | — | — | 1 | - |
| CHEMBL3957252 | — | — | 1 | - |
| CHEMBL4461552 | — | — | 1 | - |
| CHEMBL4444206 | — | — | 1 | - |
| CHEMBL4517096 | — | — | 1 | - |
| CHEMBL3941082 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4524153 | — | Ki | = | 0.16 | nM | 9.80 |
| CHEMBL4113471 | — | Ki | = | 0.8 | nM | 9.10 |
| CHEMBL4109262 | — | Ki | = | 0.9 | nM | 9.05 |
| CHEMBL4073390 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL4111969 | — | Ki | = | 1.7 | nM | 8.77 |
| CHEMBL4115120 | — | Ki | = | 3.1 | nM | 8.51 |
| CHEMBL3692392 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL3692489 | — | Ki | = | 14.0 | nM | 7.85 |
| CHEMBL3978002 | — | Ki | = | 582.0 | nM | 6.24 |
| CHEMBL4546659 | — | Ki | = | 634.0 | nM | 6.20 |
| CHEMBL3896516 | — | Ki | > | 250.0 | nM | - |
| CHEMBL3957252 | — | Ki | > | 1250.0 | nM | - |
| CHEMBL4461552 | — | Ki | > | 1250.0 | nM | - |
| CHEMBL4444206 | — | Ki | > | 1250.0 | nM | - |
| CHEMBL4517096 | — | Ki | > | 1250.0 | nM | - |
| CHEMBL3941082 | — | Ki | >= | 1250.0 | nM | - |