Assay Detail
Functional
CHEMBL4841980
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 by calcium aequorin assay
21
Total Activities
21
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
N-Terminus to Arginine Side-Chain Cyclization of Linear Peptidic Neuropeptide Y Y<sub>4</sub> Receptor Ligands Results in Picomolar Binding Constants.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 19 | 7.20 | 9.00 |
| pEC50 | 2 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4856311 | — | — | 1 | 9.00 |
| CHEMBL4873376 | — | — | 1 | 8.57 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | 2.0 | 1 | 7.96 |
| CHEMBL4857577 | — | — | 1 | 7.82 |
| CHEMBL4848958 | — | — | 1 | 7.59 |
| CHEMBL4863955 | — | — | 1 | 7.12 |
| CHEMBL4874850 | — | — | 1 | 7.04 |
| CHEMBL4870168 | — | — | 1 | 6.98 |
| CHEMBL4860290 | — | — | 1 | 6.75 |
| CHEMBL4633593 | — | — | 1 | 6.74 |
| CHEMBL4852799 | — | — | 1 | 6.72 |
| CHEMBL4865048 | — | — | 1 | 6.69 |
| CHEMBL4866086 | — | — | 1 | 6.44 |
| CHEMBL4874445 | — | — | 1 | 6.42 |
| CHEMBL4858915 | — | — | 1 | 6.17 |
| CHEMBL4862140 | — | — | 1 | - |
| CHEMBL4877802 | — | — | 1 | - |
| CHEMBL4866955 | — | — | 1 | - |
| CHEMBL4852354 | — | — | 1 | - |
| CHEMBL4868787 | — | — | 1 | - |
| CHEMBL4861544 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4856311 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4873376 | — | EC50 | = | 2.692 | nM | 8.57 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | EC50 | = | 10.96 | nM | 7.96 |
| CHEMBL4857577 | — | EC50 | = | 15.14 | nM | 7.82 |
| CHEMBL4848958 | — | EC50 | = | 25.7 | nM | 7.59 |
| CHEMBL4863955 | — | EC50 | = | 75.86 | nM | 7.12 |
| CHEMBL4874850 | — | EC50 | = | 91.2 | nM | 7.04 |
| CHEMBL4870168 | — | EC50 | = | 104.71 | nM | 6.98 |
| CHEMBL4860290 | — | EC50 | = | 177.83 | nM | 6.75 |
| CHEMBL4633593 | — | EC50 | = | 181.97 | nM | 6.74 |
| CHEMBL4852799 | — | EC50 | = | 190.55 | nM | 6.72 |
| CHEMBL4865048 | — | EC50 | = | 204.17 | nM | 6.69 |
| CHEMBL4866086 | — | EC50 | = | 363.08 | nM | 6.44 |
| CHEMBL4874445 | — | EC50 | = | 380.19 | nM | 6.42 |
| CHEMBL4858915 | — | EC50 | = | 676.08 | nM | 6.17 |
| CHEMBL4862140 | — | pEC50 | - | — | - | |
| CHEMBL4877802 | — | pEC50 | - | — | - | |
| CHEMBL4866955 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL4852354 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL4868787 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL4861544 | — | EC50 | > | 10000.0 | nM | - |