Assay Detail
Binding
CHEMBL5100327
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Inhibition of TEL-FGFR3 in mouse BaF3 cells incubated for 125 mins by plate reader analysis
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | BaF3 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of Potent and Selective Inhibitors of Wild-Type and Gatekeeper Mutant Fibroblast Growth Factor Receptor (FGFR) 2/3.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 7.64 | 8.27 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5187371 | — | — | 1 | 8.27 |
| CHEMBL5180631 | — | — | 1 | 8.26 |
| CHEMBL5203027 | — | — | 1 | 8.14 |
| CHEMBL5206837 | — | — | 1 | 7.92 |
| CHEMBL5184953 | — | — | 1 | 7.89 |
| CHEMBL5202408 | — | — | 1 | 7.85 |
| CHEMBL5200643 | — | — | 1 | 7.82 |
| CHEMBL5172121 | — | — | 1 | 7.66 |
| CHEMBL5202943 | — | — | 1 | 7.54 |
| CHEMBL5199231 | — | — | 1 | 7.54 |
| CHEMBL5201556 | — | — | 1 | 7.48 |
| CHEMBL5196280 | — | — | 1 | 7.38 |
| CHEMBL5174279 | — | — | 1 | 7.17 |
| CHEMBL5208443 | — | — | 1 | 6.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5187371 | — | IC50 | = | 5.4 | nM | 8.27 |
| CHEMBL5180631 | — | IC50 | = | 5.5 | nM | 8.26 |
| CHEMBL5203027 | — | IC50 | = | 7.2 | nM | 8.14 |
| CHEMBL5206837 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL5184953 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL5202408 | — | IC50 | = | 14.0 | nM | 7.85 |
| CHEMBL5200643 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL5172121 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL5202943 | — | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL5199231 | — | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL5201556 | — | IC50 | = | 33.0 | nM | 7.48 |
| CHEMBL5196280 | — | IC50 | = | 42.0 | nM | 7.38 |
| CHEMBL5174279 | — | IC50 | = | 68.0 | nM | 7.17 |
| CHEMBL5208443 | — | IC50 | = | 969.0 | nM | 6.01 |