Assay Detail
Binding
CHEMBL5225359
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Inhibition of p38alpha (unknown origin)
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The Emerging Landscape of Small-Molecule Therapeutics for the Treatment of Huntington's Disease.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 7.19 | 8.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5271950 | — | — | 1 | 8.12 |
| CHEMBL524174 | — | — | 1 | 7.96 |
| CHEMBL4074524 | — | — | 1 | 7.77 |
| CHEMBL5269500 | — | — | 1 | 7.62 |
| CHEMBL5284967 | — | — | 1 | 7.58 |
| CHEMBL5274433 | — | — | 1 | 7.54 |
| CHEMBL3394106 | — | — | 1 | 7.52 |
| CHEMBL5287474 | — | — | 1 | 7.47 |
| CHEMBL4077018 | — | — | 1 | 7.44 |
| CHEMBL10 | SB-203580 | — | 1 | 7.30 |
| CHEMBL426183 | — | — | 1 | 6.97 |
| CHEMBL432798 | — | — | 1 | 6.30 |
| CHEMBL313417 | — | — | 1 | 5.82 |
| CHEMBL5281537 | — | — | 1 | 5.22 |
| CHEMBL5194871 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5271950 | — | IC50 | = | 7.5 | nM | 8.12 |
| CHEMBL524174 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL4074524 | — | IC50 | = | 17.0 | nM | 7.77 |
| CHEMBL5269500 | — | IC50 | = | 24.0 | nM | 7.62 |
| CHEMBL5284967 | — | IC50 | = | 26.0 | nM | 7.58 |
| CHEMBL5274433 | — | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL3394106 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL5287474 | — | IC50 | = | 34.0 | nM | 7.47 |
| CHEMBL4077018 | — | IC50 | = | 36.0 | nM | 7.44 |
| CHEMBL10 | SB-203580 | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL426183 | — | IC50 | = | 108.0 | nM | 6.97 |
| CHEMBL432798 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL313417 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL5281537 | — | IC50 | = | 6084.0 | nM | 5.22 |
| CHEMBL5194871 | — | IC50 | > | 10000.0 | nM | - |