Assay Detail
Binding
CHEMBL5225360
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of JNK3 (unknown origin)
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The Emerging Landscape of Small-Molecule Therapeutics for the Treatment of Huntington's Disease.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 7.30 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4077018 | — | — | 1 | 9.52 |
| CHEMBL5271950 | — | — | 1 | 8.33 |
| CHEMBL3394106 | — | — | 1 | 7.75 |
| CHEMBL4074524 | — | — | 1 | 7.62 |
| CHEMBL5287474 | — | — | 1 | 7.58 |
| CHEMBL5284967 | — | — | 1 | 7.32 |
| CHEMBL5274433 | — | — | 1 | 7.13 |
| CHEMBL5281537 | — | — | 1 | 7.03 |
| CHEMBL524174 | — | — | 1 | 6.74 |
| CHEMBL5194871 | — | — | 1 | 6.74 |
| CHEMBL426183 | — | — | 1 | 6.70 |
| CHEMBL5269500 | — | — | 1 | 6.36 |
| CHEMBL10 | SB-203580 | — | 1 | 6.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4077018 | — | IC50 | = | 0.3 | nM | 9.52 |
| CHEMBL5271950 | — | IC50 | = | 4.7 | nM | 8.33 |
| CHEMBL3394106 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL4074524 | — | IC50 | = | 24.0 | nM | 7.62 |
| CHEMBL5287474 | — | IC50 | = | 26.0 | nM | 7.58 |
| CHEMBL5284967 | — | IC50 | = | 48.0 | nM | 7.32 |
| CHEMBL5274433 | — | IC50 | = | 74.0 | nM | 7.13 |
| CHEMBL5281537 | — | IC50 | = | 94.0 | nM | 7.03 |
| CHEMBL524174 | — | IC50 | = | 181.0 | nM | 6.74 |
| CHEMBL5194871 | — | IC50 | = | 184.0 | nM | 6.74 |
| CHEMBL426183 | — | IC50 | = | 202.0 | nM | 6.70 |
| CHEMBL5269500 | — | IC50 | = | 433.0 | nM | 6.36 |
| CHEMBL10 | SB-203580 | IC50 | = | 720.0 | nM | 6.14 |