Assay Detail
Binding
CHEMBL5234065
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Inhibition of USP47 (unknown origin)
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Ubiquitin carboxyl-terminal hydrolase 47 (CHEMBL2157851) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Recent advances in the development of ubiquitin-specific-processing protease 7 (USP7) inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 5.70 | 6.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2159507 | — | — | 1 | 6.46 |
| CHEMBL2398212 | — | — | 1 | 6.40 |
| CHEMBL2159505 | — | — | 1 | 6.30 |
| CHEMBL2159503 | — | — | 1 | 6.28 |
| CHEMBL2159504 | — | — | 1 | 6.06 |
| CHEMBL2159500 | — | — | 1 | 5.92 |
| CHEMBL2159501 | — | — | 1 | 5.89 |
| CHEMBL2159499 | — | — | 1 | 5.66 |
| CHEMBL4569978 | — | — | 1 | 5.46 |
| CHEMBL5281075 | — | — | 1 | 5.37 |
| CHEMBL2159502 | — | — | 1 | 5.26 |
| CHEMBL2159496 | — | — | 1 | 4.85 |
| CHEMBL5283229 | — | — | 1 | 4.18 |
| CHEMBL4516637 | — | — | 1 | - |
| CHEMBL5274053 | — | — | 1 | - |
| CHEMBL5276519 | — | — | 1 | - |
| CHEMBL5270413 | — | — | 1 | - |
| CHEMBL4438288 | — | — | 1 | - |
| CHEMBL5286198 | — | — | 1 | - |
| CHEMBL5277194 | — | — | 1 | - |
| CHEMBL2159506 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2159507 | — | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL2398212 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL2159505 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL2159503 | — | IC50 | = | 530.0 | nM | 6.28 |
| CHEMBL2159504 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL2159500 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL2159501 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL2159499 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL4569978 | — | IC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL5281075 | — | IC50 | = | 4300.0 | nM | 5.37 |
| CHEMBL2159502 | — | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL2159496 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL5283229 | — | IC50 | = | 66000.0 | nM | 4.18 |
| CHEMBL4516637 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5274053 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5276519 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5270413 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4438288 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5286198 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5277194 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2159506 | — | IC50 | > | 31600.0 | nM | - |