Assay Detail
Binding
CHEMBL5376120
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Agonist activity at MRGPRX4 83L (unknown origin) expressed in CHO cells assessed as induction of beta-arrestin recruitment measured after 90 mins by luminescence assay
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery of Potent Agonists for the Predominant Variant of the Orphan MAS-Related G Protein-Coupled Receptor X4 (MRGPRX4).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 25 | 5.11 | 6.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5402204 | — | — | 1 | 6.26 |
| CHEMBL5408931 | — | — | 1 | 5.41 |
| CHEMBL783 | NATEGLINIDE | 4.0 | 1 | 5.39 |
| CHEMBL5420073 | — | — | 1 | 5.24 |
| CHEMBL5408226 | — | — | 1 | 5.20 |
| CHEMBL5403433 | — | — | 1 | 5.17 |
| CHEMBL406393 | DEOXYCHOLIC ACID | 4.0 | 1 | 4.61 |
| CHEMBL1551 | URSODIOL | 4.0 | 1 | 4.47 |
| CHEMBL412272 | TAURODEOXYCHOLIC ACID | 2.0 | 1 | 4.25 |
| CHEMBL1205720 | — | — | 1 | - |
| CHEMBL5394109 | — | — | 1 | - |
| CHEMBL5400164 | — | — | 1 | - |
| CHEMBL5394574 | — | — | 1 | - |
| CHEMBL5418196 | — | — | 1 | - |
| CHEMBL5411533 | — | — | 1 | - |
| CHEMBL5427570 | — | — | 1 | - |
| CHEMBL5416729 | — | — | 1 | - |
| CHEMBL5439076 | — | — | 1 | - |
| CHEMBL5427296 | — | — | 1 | - |
| CHEMBL5424935 | — | — | 1 | - |
| CHEMBL5434279 | — | — | 1 | - |
| CHEMBL5403197 | — | — | 1 | - |
| CHEMBL5432461 | — | — | 1 | - |
| CHEMBL5428142 | — | — | 1 | - |
| CHEMBL5425100 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5402204 | — | EC50 | = | 548.0 | nM | 6.26 |
| CHEMBL5408931 | — | EC50 | = | 3940.0 | nM | 5.41 |
| CHEMBL783 | NATEGLINIDE | EC50 | = | 4090.0 | nM | 5.39 |
| CHEMBL5420073 | — | EC50 | = | 5710.0 | nM | 5.24 |
| CHEMBL5408226 | — | EC50 | = | 6280.0 | nM | 5.20 |
| CHEMBL5403433 | — | EC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL406393 | DEOXYCHOLIC ACID | EC50 | = | 24600.0 | nM | 4.61 |
| CHEMBL1551 | URSODIOL | EC50 | = | 33800.0 | nM | 4.47 |
| CHEMBL412272 | TAURODEOXYCHOLIC ACID | EC50 | = | 55700.0 | nM | 4.25 |
| CHEMBL1205720 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5394109 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5400164 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5394574 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5418196 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5411533 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5427570 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5416729 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5439076 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5427296 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5424935 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5434279 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5403197 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5432461 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5428142 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5425100 | — | EC50 | > | 10000.0 | nM | - |