Assay Detail
Functional
CHEMBL5524108
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Agonist activity at human FPR2
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The formyl peptide receptors FPR1 and FPR2 as targets for inflammatory disorders: recent advances in the development of small-molecule agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 10 | 8.93 | 10.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL552527 | — | — | 1 | 10.15 |
| CHEMBL5287715 | — | — | 1 | 9.60 |
| CHEMBL4784510 | BMS-986235 | 1.0 | 1 | 9.39 |
| CHEMBL5286212 | — | — | 1 | 9.18 |
| CHEMBL5564062 | — | — | 1 | 8.92 |
| CHEMBL5555475 | — | — | 1 | 8.62 |
| CHEMBL5560735 | — | — | 1 | 8.42 |
| CHEMBL5282051 | — | — | 1 | 8.39 |
| CHEMBL379761 | — | — | 1 | 7.66 |
| CHEMBL564392 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL552527 | — | EC50 | = | 0.07 | nM | 10.15 |
| CHEMBL5287715 | — | EC50 | = | 0.25 | nM | 9.60 |
| CHEMBL4784510 | BMS-986235 | EC50 | = | 0.41 | nM | 9.39 |
| CHEMBL5286212 | — | EC50 | = | 0.66 | nM | 9.18 |
| CHEMBL5564062 | — | EC50 | = | 1.2 | nM | 8.92 |
| CHEMBL5555475 | — | EC50 | = | 2.4 | nM | 8.62 |
| CHEMBL5560735 | — | EC50 | = | 3.8 | nM | 8.42 |
| CHEMBL5282051 | — | EC50 | = | 4.1 | nM | 8.39 |
| CHEMBL379761 | — | EC50 | = | 22.0 | nM | 7.66 |
| CHEMBL564392 | — | EC50 | > | 50.0 | nM | - |