Assay Detail
Binding
CHEMBL640329
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Binding affinity for [125I]AB-MECA against rat Adenosine A3 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Synthesis and biological activities of flavonoid derivatives as A3 adenosine receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 4.83 | 4.91 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL76874 | — | — | 1 | 4.91 |
| CHEMBL72862 | — | — | 1 | 4.74 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL76874 | — | Ki | = | 12300.0 | nM | 4.91 |
| CHEMBL72862 | — | Ki | = | 18200.0 | nM | 4.74 |