Assay Detail
Functional
CHEMBL885178
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Concentration required to inhibit dexamethasone-induced death of mice thymocytes
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Inhibitors of apoptosis in lymphocytes: synthesis and biological evaluation of compounds related to pifithrin-alpha.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 26 | 5.39 | 6.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL194367 | — | — | 1 | 6.46 |
| CHEMBL130474 | — | — | 1 | 5.91 |
| CHEMBL371682 | — | — | 1 | 5.88 |
| CHEMBL196147 | — | — | 1 | 5.74 |
| CHEMBL193504 | — | — | 1 | 5.70 |
| CHEMBL382067 | — | — | 1 | 5.64 |
| CHEMBL196846 | — | — | 1 | 5.42 |
| CHEMBL382727 | — | — | 1 | 5.40 |
| CHEMBL196158 | — | — | 1 | 5.40 |
| CHEMBL198759 | — | — | 1 | 5.38 |
| CHEMBL362918 | — | — | 1 | 5.35 |
| CHEMBL370909 | — | — | 1 | 5.32 |
| CHEMBL198196 | — | — | 1 | 5.27 |
| CHEMBL440568 | — | — | 1 | 5.25 |
| CHEMBL381199 | — | — | 1 | 5.24 |
| CHEMBL194798 | — | — | 1 | 5.22 |
| CHEMBL199083 | — | — | 1 | 5.14 |
| CHEMBL194973 | — | — | 1 | 5.14 |
| CHEMBL198633 | — | — | 1 | 5.12 |
| CHEMBL370460 | — | — | 1 | 5.09 |
| CHEMBL199257 | — | — | 1 | 5.01 |
| CHEMBL199092 | — | — | 1 | 5.01 |
| CHEMBL129256 | — | — | 1 | 4.99 |
| CHEMBL381036 | — | — | 1 | - |
| CHEMBL197575 | — | — | 1 | - |
| CHEMBL194638 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL194367 | — | EC50 | = | 350.0 | nM | 6.46 |
| CHEMBL130474 | — | EC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL371682 | — | EC50 | = | 1310.0 | nM | 5.88 |
| CHEMBL196147 | — | EC50 | = | 1840.0 | nM | 5.74 |
| CHEMBL193504 | — | EC50 | = | 2010.0 | nM | 5.70 |
| CHEMBL382067 | — | EC50 | = | 2290.0 | nM | 5.64 |
| CHEMBL196846 | — | EC50 | = | 3790.0 | nM | 5.42 |
| CHEMBL382727 | — | EC50 | = | 4020.0 | nM | 5.40 |
| CHEMBL196158 | — | EC50 | = | 4020.0 | nM | 5.40 |
| CHEMBL198759 | — | EC50 | = | 4160.0 | nM | 5.38 |
| CHEMBL362918 | — | EC50 | = | 4440.0 | nM | 5.35 |
| CHEMBL370909 | — | EC50 | = | 4770.0 | nM | 5.32 |
| CHEMBL198196 | — | EC50 | = | 5370.0 | nM | 5.27 |
| CHEMBL440568 | — | EC50 | = | 5680.0 | nM | 5.25 |
| CHEMBL381199 | — | EC50 | = | 5720.0 | nM | 5.24 |
| CHEMBL194798 | — | EC50 | = | 6060.0 | nM | 5.22 |
| CHEMBL199083 | — | EC50 | = | 7260.0 | nM | 5.14 |
| CHEMBL194973 | — | EC50 | = | 7280.0 | nM | 5.14 |
| CHEMBL198633 | — | EC50 | = | 7540.0 | nM | 5.12 |
| CHEMBL370460 | — | EC50 | = | 8120.0 | nM | 5.09 |
| CHEMBL199257 | — | EC50 | = | 9690.0 | nM | 5.01 |
| CHEMBL199092 | — | EC50 | = | 9840.0 | nM | 5.01 |
| CHEMBL129256 | — | EC50 | = | 10230.0 | nM | 4.99 |
| CHEMBL381036 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL197575 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL194638 | — | EC50 | > | 10000.0 | nM | - |