Assay Detail
Functional
CHEMBL906537
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Inhibition of fMLP-induced superoxide production in human neutrophils
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Neutrophil |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Anti-inflammatory benzenoids from Antrodia camphorata.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 4.59 | 5.07 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL388526 | ANTICIN A | — | 1 | 5.07 |
| CHEMBL229169 | ANTROCAMPHIN A | — | 1 | 5.03 |
| CHEMBL446448 | ANTCIN B | — | 1 | 5.01 |
| CHEMBL229343 | — | — | 1 | 4.58 |
| CHEMBL521 | IBUPROFEN | 4.0 | 1 | 4.56 |
| CHEMBL426367 | EBURICOL | — | 1 | 4.30 |
| CHEMBL1744446 | DEHYDROEBURICOIC ACID | — | 1 | 4.11 |
| CHEMBL252915 | SESAMIN | — | 1 | 4.04 |
| CHEMBL221543 | BETA-SITOSTENONE | — | 1 | - |
| CHEMBL229618 | — | — | 1 | - |
| CHEMBL229563 | — | — | 1 | - |
| CHEMBL229509 | — | — | 1 | - |
| CHEMBL229460 | ANTRODIOXOLANONE | — | 1 | - |
| CHEMBL376803 | — | — | 1 | - |
| CHEMBL229342 | ANTROCAMPHIN B | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL388526 | ANTICIN A | IC50 | = | 8550.0 | nM | 5.07 |
| CHEMBL229169 | ANTROCAMPHIN A | IC50 | = | 9330.0 | nM | 5.03 |
| CHEMBL446448 | ANTCIN B | IC50 | = | 9820.0 | nM | 5.01 |
| CHEMBL229343 | — | IC50 | = | 26090.0 | nM | 4.58 |
| CHEMBL521 | IBUPROFEN | IC50 | = | 27500.0 | nM | 4.56 |
| CHEMBL426367 | EBURICOL | IC50 | = | 50470.0 | nM | 4.30 |
| CHEMBL1744446 | DEHYDROEBURICOIC ACID | IC50 | = | 77500.0 | nM | 4.11 |
| CHEMBL252915 | SESAMIN | IC50 | = | 90230.0 | nM | 4.04 |
| CHEMBL221543 | BETA-SITOSTENONE | IC50 | > | 100000.0 | nM | - |
| CHEMBL229618 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL229563 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL229509 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL229460 | ANTRODIOXOLANONE | IC50 | > | 100000.0 | nM | - |
| CHEMBL376803 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL229342 | ANTROCAMPHIN B | IC50 | > | 100000.0 | nM | - |