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Compound Detail

CHEMBL150457

p-Xyloquinone
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CC1=CC(=O)C(C)=CC1=O

Basic Information

ChEMBL ID CHEMBL150457
Name p-Xyloquinone
Phase Preclinical
Structure Type MOL
InChI Key MYKLQMNSFPAPLZ-UHFFFAOYSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
13
Publications
0
Known Names

Molecular Properties

136.2
MW (Da)
1.03
ALogP
2
HBA
0
HBD
34.1
PSA (Ų)
0.47
QED
0
Ro5 Violations
0
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C8H8O2
MW 136.15
Aromatic Rings 0
Heavy Atoms 10
NP-Likeness 0.98

Activity Summary

IC50 2 meas. best 6.19

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
HL-60
CHEMBL383
IC50 6.19 6.19 640.0 1
K562
CHEMBL385
IC50 6.12 6.12 750.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
HL-60 IC50 = 640.0 nM 6.19 Antiproliferative activity against human HL60 cells 18052030
K562 IC50 = 750.0 nM 6.12 In vitro cytotoxicity against Human Chronic Leukemia K562 cells 8558523

Literature References

PubMed DOI Target Context # Activities
18461966 10.1021/jf800331r Coptotermes formosanus 4
8558523 10.1021/jm950629q Nucleic Acid 2
8576915 10.1021/jm9405147 No relevant target 2
8558523 10.1021/jm950629q K562 1
8576915 10.1021/jm9405147 ADMET 1
18052030 10.1021/np070436t HL-60 1
1710653 10.1021/np50073a012 Human immunodeficiency virus type 1 reverse transcriptase 1
20851600 10.1016/j.bmcl.2010.08.129 Candida albicans 1
20851600 10.1016/j.bmcl.2010.08.129 Candida tropicalis 1
20851600 10.1016/j.bmcl.2010.08.129 Pichia kudriavzevii 1
20851600 10.1016/j.bmcl.2010.08.129 Cryptococcus neoformans 1
20851600 10.1016/j.bmcl.2010.08.129 Aspergillus niger 1
20851600 10.1016/j.bmcl.2010.08.129 Aspergillus flavus 1

Data from ChEMBL 36 via Core Engine