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Compound Detail

CHEMBL373719

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COc1ccc(C(=O)NN2C(=O)[C@@H]3C4C=CC(C5CC54)[C@@H]3C2=O)cc1

Basic Information

ChEMBL ID CHEMBL373719
Phase Preclinical
Structure Type MOL
InChI Key ZPZCRHNAIUYXKE-YOHVKPHQSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

338.4
MW (Da)
1.39
ALogP
4
HBA
1
HBD
75.7
PSA (Ų)
0.67
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H18N2O4
MW 338.36
Aromatic Rings 1
Heavy Atoms 25
NP-Likeness -0.40

Activity Summary

EC50 2 meas. best 5.66

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Vaccinia virus
CHEMBL613493
EC50 5.66 5.66 2200.0 1
Cowpox virus
CHEMBL612672
EC50 5.51 5.51 3100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
17335190 10.1021/jm061484y Cowpox virus 2
17335190 10.1021/jm061484y Vaccinia virus 1
17335190 10.1021/jm061484y ADMET 1

Data from ChEMBL 36 via Core Engine