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Compound Detail

CHEMBL373720

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Cn1cccc1C(=O)NN1C(=O)[C@@H]2C3C=CC(C4CC43)[C@@H]2C1=O

Basic Information

ChEMBL ID CHEMBL373720
Phase Preclinical
Structure Type MOL
InChI Key KMIXNGXFOCHOTL-UHPCZEEKSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

311.3
MW (Da)
0.72
ALogP
4
HBA
1
HBD
71.4
PSA (Ų)
0.65
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C17H17N3O3
MW 311.34
Aromatic Rings 1
Heavy Atoms 23
NP-Likeness -0.68

Activity Summary

EC50 2 meas. best 5.33

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Cowpox virus
CHEMBL612672
EC50 5.33 5.33 4700.0 1
Vaccinia virus
CHEMBL613493
EC50 4.8 4.8 15800.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
17335190 10.1021/jm061484y Cowpox virus 2
17335190 10.1021/jm061484y Vaccinia virus 1
17335190 10.1021/jm061484y ADMET 1

Data from ChEMBL 36 via Core Engine