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Compound Detail

CHEMBL4520626

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O=C(NC(=S)NNC(=O)c1ccc(O)cc1O)c1ccccc1

Basic Information

ChEMBL ID CHEMBL4520626
Phase Preclinical
Structure Type MOL
InChI Key XONNGRHIIOMDMC-UHFFFAOYSA-N
2
Targets
2
Activities
2
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

331.4
MW (Da)
1.05
ALogP
5
HBA
5
HBD
110.7
PSA (Ų)
0.42
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C15H13N3O4S
MW 331.35
Aromatic Rings 2
Heavy Atoms 23
NP-Likeness -1.23

Activity Summary

EC50 1 meas. best 5.9
Ki 1 meas. best 5.9

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Synechocystis sp. PCC 6803
CHEMBL4513211
EC50 5.9 5.9 1250.0 1
Fructose-bisphosphate aldolase class 2
CHEMBL4523320
Ki 5.9 5.9 1250.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
30711311 10.1016/j.bmc.2019.01.023 Synechocystis sp. PCC 6803 1
30711311 10.1016/j.bmc.2019.01.023 Fructose-bisphosphate aldolase class 2 1

Data from ChEMBL 36 via Core Engine