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Compound Detail

CHEMBL56723

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CN(C)c1cc(O)nc(N)n1

Basic Information

ChEMBL ID CHEMBL56723
Phase Preclinical
Structure Type MOL
InChI Key KCSATFXTZGNTPK-UHFFFAOYSA-N
3
Targets
3
Activities
1
Assay Types
0
PK Parameters
8
Publications
0
Known Names

Molecular Properties

154.2
MW (Da)
-0.17
ALogP
5
HBA
2
HBD
75.3
PSA (Ų)
0.59
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C6H10N4O
MW 154.17
Aromatic Rings 1
Heavy Atoms 11
NP-Likeness -1.32

Activity Summary

IC50 3 meas. best 9.49

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human alphaherpesvirus 3
CHEMBL613132
IC50 9.49 9.49 0.3 1
Human alphaherpesvirus 2
CHEMBL370
IC50 8.59 8.59 2.6 1
Human alphaherpesvirus 1
CHEMBL377
IC50 8.59 8.59 2.6 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
11960502 10.1021/jm011095y E6SM 3
11960502 10.1021/jm011095y HEL 3
11960502 10.1021/jm011095y CCRF-CEM 2
11960502 10.1021/jm011095y Human alphaherpesvirus 3 1
11960502 10.1021/jm011095y Moloney murine sarcoma virus 1
19112024 10.1016/j.bmc.2008.11.075 Human alphaherpesvirus 1 1
19112024 10.1016/j.bmc.2008.11.075 Human alphaherpesvirus 2 1
19112024 10.1016/j.bmc.2008.11.075 Human alphaherpesvirus 3 1

Data from ChEMBL 36 via Core Engine