Assay Detail
Binding
CHEMBL1613879
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for HCV NS3 helicase inhibitors: Fluorescence-based biochemical high-throughput dose response assay for compounds that cause fluorescent intercalator displacement (FID). (Class of assay: confirmatory) [Related pubchem assays: 1830 (Summary AID.), 1945 (Screening assay (Fluorescence-based displacement)), 1800 (Counterscreen (NS3 inhibitors).)]
125
Total Activities
125
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 125 | 4.42 | 4.65 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1493191 | — | — | 1 | 4.65 |
| CHEMBL1495335 | — | — | 1 | 4.55 |
| CHEMBL1589514 | — | — | 1 | 4.54 |
| CHEMBL1580969 | — | — | 1 | 4.52 |
| CHEMBL1347122 | — | — | 1 | 4.49 |
| CHEMBL1543865 | — | — | 1 | 4.47 |
| CHEMBL1546396 | — | — | 1 | 4.30 |
| CHEMBL1545427 | — | — | 1 | 4.14 |
| CHEMBL1500600 | — | — | 1 | 4.08 |
| CHEMBL1527520 | — | — | 1 | - |
| CHEMBL1576217 | — | — | 1 | - |
| CHEMBL1605561 | — | — | 1 | - |
| CHEMBL1576490 | — | — | 1 | - |
| CHEMBL1449425 | — | — | 1 | - |
| CHEMBL1605743 | — | — | 1 | - |
| CHEMBL1595235 | — | — | 1 | - |
| CHEMBL1371074 | — | — | 1 | - |
| CHEMBL1301164 | — | — | 1 | - |
| CHEMBL1991888 | — | — | 1 | - |
| CHEMBL1537336 | — | — | 1 | - |
| CHEMBL1536896 | — | — | 1 | - |
| CHEMBL1299903 | — | — | 1 | - |
| CHEMBL1399109 | — | — | 1 | - |
| CHEMBL3192400 | — | — | 1 | - |
| CHEMBL1594488 | — | — | 1 | - |
| CHEMBL1458120 | — | — | 1 | - |
| CHEMBL1438291 | — | — | 1 | - |
| CHEMBL1299566 | — | — | 1 | - |
| CHEMBL1594376 | — | — | 1 | - |
| CHEMBL1447158 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1493191 | — | IC50 | = | 22278.0 | nM | 4.65 |
| CHEMBL1495335 | — | IC50 | = | 28026.0 | nM | 4.55 |
| CHEMBL1589514 | — | IC50 | = | 28890.0 | nM | 4.54 |
| CHEMBL1580969 | — | IC50 | = | 30467.0 | nM | 4.52 |
| CHEMBL1347122 | — | IC50 | = | 32288.0 | nM | 4.49 |
| CHEMBL1543865 | — | IC50 | = | 33757.0 | nM | 4.47 |
| CHEMBL1546396 | — | IC50 | = | 49740.0 | nM | 4.30 |
| CHEMBL1545427 | — | IC50 | = | 72227.0 | nM | 4.14 |
| CHEMBL1500600 | — | IC50 | = | 83505.0 | nM | 4.08 |
| CHEMBL1334412 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1486503 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1437673 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1492622 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1563898 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1366482 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1562843 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1546228 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL3198103 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1496459 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL599013 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1549566 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL3195767 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1587849 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1587715 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1446502 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1587683 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1448067 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL3195976 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1509648 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1387693 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1389429 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1504875 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1364584 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL3197424 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1489865 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1544163 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1347385 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1337304 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1982808 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1561333 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1584828 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL602213 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1544885 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1365290 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1387835 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1600566 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1378059 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL3196732 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1444743 | — | IC50 | > | 79365.0 | nM | - |
| CHEMBL1338595 | — | IC50 | > | 79365.0 | nM | - |