Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL1563898

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
O=c1cc2oc3cc(O)c(O)cc3c(-c3ccccc3[N+](=O)[O-])c-2cc1O

Basic Information

ChEMBL ID CHEMBL1563898
Phase Preclinical
Structure Type MOL
InChI Key ZULBKXYQNMBEJG-UHFFFAOYSA-N
9
Targets
15
Activities
2
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

365.3
MW (Da)
3.59
ALogP
7
HBA
3
HBD
134.0
PSA (Ų)
0.21
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H11NO7
MW 365.30
Aromatic Rings 2
Heavy Atoms 27
NP-Likeness 0.43

Activity Summary

EC50 8 meas. best 5.97
IC50 7 meas. best 6.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NS3
CHEMBL1293269
IC50 6.0 6.0 990.0 1
Unchecked
CHEMBL612545
EC50 5.97 5.3433 1073.0 3
ATP-dependent molecular chaperone HSP82
CHEMBL1293251
EC50 5.82 5.82 1522.0 1
Troponin, cardiac muscle
CHEMBL2095202
IC50 5.79 5.79 1640.0 1
Unchecked
CHEMBL612545
IC50 5.14 4.6433 7230.0 3
Streptococcus sp. 'group A'
CHEMBL612389
EC50 5.1 5.1 7937.0 1
Streptokinase A
CHEMBL1293228
EC50 5.03 4.99 9355.0 2
Streptococcus
CHEMBL612313
EC50 4.99 4.99 10172.0 1
Matrix metalloproteinase-14
CHEMBL3869
IC50 4.75 4.75 17900.0 1
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1
CHEMBL3964
IC50 4.17 4.17 67500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
NS3 IC50 = 990.0 nM 6.0 PUBCHEM_BIOASSAY: Fluorescence-based biochemical high throughput dose response a... -
Unchecked EC50 = 1073.0 nM 5.97 PUBCHEM_BIOASSAY: Fluorescence Cell-Based Retest of Candida albicans Growth in t... -
ATP-dependent molecular chaperone HSP82 EC50 = 1522.0 nM 5.82 PUBCHEM_BIOASSAY: Fluorescence Cell-Based Secondary Assay to Identify Inhibitors... -
Troponin, cardiac muscle IC50 = 1640.0 nM 5.79 PUBCHEM_BIOASSAY: Fluorescence-based biochemical high throughput dose response a... -
Unchecked IC50 = 7230.0 nM 5.14 PUBCHEM_BIOASSAY: A biochemical assay using the ADP-Hunter methodology, purified... -
Streptococcus sp. 'group A' EC50 = 7937.0 nM 5.1 PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Confirmation HTS to Iden... -
Unchecked EC50 = 8253.0 nM 5.08 PUBCHEM_BIOASSAY: Fluorescence Cell-Based Secondary Assay for toxicity in mammal... -
Streptokinase A EC50 = 9355.0 nM 5.03 PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Confirmation HTS to Iden... -
Streptococcus EC50 = 10172.0 nM 4.99 PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Response HTS to Identify... -
Unchecked EC50 = 10500.0 nM 4.98 PUBCHEM_BIOASSAY: A cytotoxicity screen of small molecule inhibitors of the PhoP... -
Streptokinase A EC50 = 11193.0 nM 4.95 PUBCHEM_BIOASSAY: Absorbance Microorganism-Based Dose Response HTS to Identify I... -
Matrix metalloproteinase-14 IC50 = 17900.0 nM 4.75 PubChem BioAssay. Dose Response confirmation of uHTS hits for a small molecule i... -
Unchecked IC50 = 28500.0 nM 4.54 PUBCHEM_BIOASSAY: A Counter Screen to identiry small molecule screen for inhibit... -
Unchecked IC50 = 56570.0 nM 4.25 PUBCHEM_BIOASSAY: A screen for inhibitors of the PhoP region in Salmonella Typhi... -
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1 IC50 = 67500.0 nM 4.17 PubChem BioAssay. Counterscreen for inhibitors of phospholipase C isozymes (PLC-... -

Data from ChEMBL 36 via Core Engine